SCHEMBL1709392

SCHEMBL1709392

COC(=O)C[C@H]1CCC[C@@H](NCc2ccc(C(F)(F)F)cc2)[C@@H]1c1ccc(C(F)(F)F)cc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.44
KDM1A O60341 1/20 0.42
MAOB P27338 1/20 0.42
CCR2 P41597 6/20 0.42
TACR1 P25103 4/20 0.41
SSTR3 P32745 3/20 0.40
TEAD1 P28347 1/20 0.40
KCNH2 Q12809 1/20 0.38
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
MAPK1 P28482 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
P2RX7 Q99572 1/20 0.36
KCNQ3 O43525 1/20 0.36
KCNQ2 O43526 1/20 0.36
KCNQ4 P56696 1/20 0.36
KCNQ5 Q9NR82 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1709391 0.96 SSTR3 (0.46) MAOAKDM1AMAOBCCR2TACR1
SCHEMBL1709386 0.95 MAOA (0.48) MAOAKDM1AMAOBCCR2TACR1
SCHEMBL1709387 0.83 SSTR3 (0.44) MAOAKDM1AMAOBSSTR3KDM4E
SCHEMBL1709388 0.81 MAOA (0.45) MAOAKDM1AMAOBTACR1KCNH2
SCHEMBL1709396 0.77 ALDH1A1 (0.38) TACR1KCNH2KDM4EALDH1A1GAA
SCHEMBL4495364 0.76 CCR2 (0.47) MAOAKDM1AMAOBCCR2SSTR3
SCHEMBL4481286 0.76 CCR2 (0.47) MAOAKDM1AMAOBCCR2SSTR3
SCHEMBL10033002 0.75 SLC6A2 (0.37) TACR1KCNH2KDM4EALDH1A1POLB
SCHEMBL1709467 0.75 TACR1 (0.41) TACR1KCNH2
SCHEMBL1709470 0.74 KDM4E (0.40) KDM4EALDH1A1POLBGAAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012046771-A1 CYCLOALKANE COMPOUND アステラス製薬株式会社 (JP) 2012-04-12 WO disclosed