SCHEMBL1709412

SCHEMBL1709412

C=C(O)C[C@@H]1CC[C@@H](N(CCC2CCCCC2)CC2CCCCC2)[C@H](c2ccccc2F)C1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.31
OPRK1 P41145 2/20 0.31
BCHE P06276 3/20 0.31
ACHE P22303 1/20 0.31
KDM1A O60341 4/20 0.31
KDM1B Q8NB78 1/20 0.31
HTR2C P28335 1/20 0.30
HTR2B P41595 1/20 0.30
KDM4E B2RXH2 1/20 0.30
GAA P10253 1/20 0.30
OPRL1 P41146 1/20 0.30
MAOA P21397 2/20 0.30
MAOB P27338 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10032986 0.93 KDM1A (0.34) OPRM1OPRK1KDM1AKDM1BHTR2C
SCHEMBL10033139 0.84 SIGMAR1 (0.39) KDM1AHTR2CMAOAMAOB
SCHEMBL10033179 0.83 ALDH1A1 (0.40) BCHEACHE
SCHEMBL10033140 0.81 OPRM1 (0.32) OPRM1OPRK1HTR2CHTR2BOPRL1
SCHEMBL1709491 0.81 KDM1A (0.42) BCHEACHEKDM1AMAOAMAOB
SCHEMBL1709450 0.80 HTR2C (0.33) KDM1AHTR2CMAOAMAOB
SCHEMBL10032822 0.80 HTR2C (0.33) KDM1AHTR2CMAOAMAOB
SCHEMBL1709420 0.78 SIGMAR1 (0.40) KDM1AHTR2CHTR2BMAOAMAOB
SCHEMBL10032995 0.77 HTR2A (0.34) BCHEACHEKDM1AHTR2CHTR2B
SCHEMBL10033138 0.76 SIGMAR1 (0.42) KDM1AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012046771-A1 CYCLOALKANE COMPOUND アステラス製薬株式会社 (JP) 2012-04-12 WO disclosed