SCHEMBL17101772

SCHEMBL17101772

O=S(=O)(NCc1ccc(B(O)O)cc1)c1ccccc1Cl

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.52
SLC12A2 P55011 1/20 0.52
SLC12A5 Q9H2X9 1/20 0.52
HSD11B1 P28845 1/20 0.51
GLA P06280 1/20 0.48
CA12 O43570 3/20 0.48
CA9 Q16790 3/20 0.48
NR3C2 P08235 1/20 0.47
TP53 P04637 1/20 0.47
ALDH1A1 P00352 3/20 0.46
KEAP1 Q14145 1/20 0.45
POLB P06746 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MCL1 Q07820 1/20 0.43
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17101682 0.83 LMNA (0.51) LMNACA12CA9NR3C2KEAP1
SCHEMBL17101701 0.83 NR3C2 (0.48) LMNACA12CA9NR3C2TP53
SCHEMBL5167263 0.80 SMN1; SMN2 (0.56) LMNACA12CA9ALDH1A1L3MBTL1
SCHEMBL17101697 0.80 NPY1R (0.51) LMNACA12CA9ALDH1A1KEAP1
SCHEMBL17101699 0.77 LMNA (0.47) LMNANR3C2TP53ALDH1A1MCL1
SCHEMBL17101815 0.77 LMNA (0.43) LMNACA12CA9KEAP1L3MBTL1
SCHEMBL17101704 0.77 ALDH1A1 (0.61) LMNAHSD11B1CA12CA9TP53
SCHEMBL17101822 0.76 HSD11B1 (0.61) LMNAHSD11B1TP53ALDH1A1L3MBTL1
SCHEMBL5651347 0.76 KEAP1 (0.74) LMNASLC12A2SLC12A5CA12CA9
SCHEMBL23603320 0.74 LMNA (0.56) LMNASLC12A2SLC12A5HSD11B1GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015140566-A1 PYRAZOLO-PYRIMIDINES AS INHIBITORS OF BTK REDX PHARMA PLC (GB) 2015-09-24 WO disclosed