SCHEMBL17144343

SCHEMBL17144343

COC(=O)c1ccc(Cl)c(Cl)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 3/20 0.46
MAPK1 P28482 1/20 0.46
CYP1A2 P05177 2/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
TP53 P04637 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MAPT P10636 2/20 0.43
NQO2 P16083 3/20 0.41
ALDH1A1 P00352 2/20 0.41
GAA P10253 1/20 0.41
RECQL P46063 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
PTGER4 P35408 1/20 0.40
MRGPRX4 Q96LA9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30405765 1.00 NOTUM (0.46) NOTUMMAPK1CYP1A2NPC1RAB9A
SCHEMBL2255434 0.83 SMN1; SMN2 (0.46) NOTUMMAPK1CYP1A2NPC1RAB9A
SCHEMBL16372354 0.83 LCK (0.46) NOTUMMAPK1CYP1A2NPC1RAB9A
SCHEMBL31500498 0.83 SMN1; SMN2 (0.46) NOTUMMAPK1CYP1A2NPC1RAB9A
SCHEMBL31661385 0.83 NOTUM (0.45) NOTUMMAPK1CYP1A2NPC1RAB9A
SCHEMBL1615811 0.83 NPC1 (0.46) MAPK1CYP1A2NPC1RAB9ATP53
SCHEMBL18725355 0.83 SMN1; SMN2 (0.46) NOTUMMAPK1CYP1A2NPC1RAB9A
SCHEMBL30093142 0.83 LCK (0.46) NOTUMMAPK1CYP1A2NPC1RAB9A
SCHEMBL2593348 0.81 PTPN1 (0.50) NOTUMMAPK1CYP1A2NPC1RAB9A
SCHEMBL7236303 0.81 CTSA (0.48) NOTUMMAPK1CYP1A2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 38 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4615573-A1 GLUCAGON-LIKE PEPTIDE 1 RECEPTOR AGONISTS Eli Lilly and Company (US) 2025-09-17 EP disclosed
US-20250092033-A1 HETEROAROMATIC NITROGEN-OXIDE COMPOUND, PREPARATION METHOD THEREFOR, AND USE THEREOF Beijing Avistone Biotechnology Co., Ltd. (CN) 2025-03-20 US disclosed
US-20240368122-A1 JAK2 INHIBITORS AND METHODS OF USE THEREOF RELAY THERAPEUTICS INC (US) 2024-11-07 US disclosed
EP-4458818-A1 HETEROAROMATIC NITROGEN-OXIDE COMPOUND, PREPARATION METHOD THEREFOR, AND USE THEREOF Beijing Avistone Biotechnology Co., Ltd. (CN) 2024-11-06 EP disclosed
EP-4387964-A1 JAK2 INHIBITORS AND METHODS OF USE THEREOF Relay Therapeutics, Inc. (US) 2024-06-26 EP disclosed
WO-2024102625-A1 GLUCAGON-LIKE PEPTIDE 1 RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2024-05-16 WO disclosed
US-20240083908-A1 TETRAHYDROTHIENOPYRIMIDINESULFONAMIDE COMPOUNDS ALIVEXIS, INC. (JP) 2024-03-14 US disclosed
CN-116003406-B Heteroaryl ring nitroxide compound and preparation method and application thereof 北京鞍石生物科技有限责任公司 2024-01-23 CN disclosed
EP-4269415-A1 TETRAHYDRO THIENOPYRIDINE SULFONAMIDE COMPOUND Modulus Discovery, Inc. (JP) 2023-11-01 EP disclosed
CN-116583286-A Tetrahydrothienopyrimidine sulfonamide compounds 某久拉斯株式会社 2023-08-11 CN disclosed
US-20160376262-A1 NOVEL PYRIDINE DERIVATIVES HOFFMANN-LA ROCHE INC. (US) 2016-12-29 US disclosed
WO-2016191245-A1 RECOVERY AND/OR REUSE OF PALLADIUM CATALYST AFTER A SUZUKI COUPLING DOW AGROSCIENCES LLC (US) 2016-12-01 WO disclosed
US-20160340311-A1 RECOVERY AND/OR REUSE OF PALLADIUM CATALYST AFTER A SUZUKI COUPLING DOW AGROSCIENCES LLC (US) 2016-11-24 US disclosed
CN-106132958-A Pyridine 2 amides compound as CB2 agonist 豪夫迈·罗氏有限公司 2016-11-16 CN disclosed
CN-105377830-A 4-amino-6-(heterocyclic)picolinates and 6-amino-2-(heterocyclic) pyrimidine-4-carboxylates and their use as herbicides DOW AGROSCIENCES LLC 2016-03-02 CN disclosed
CN-105209451-A 4-amino-6- (heterocyclyl) pyridine-2-carboxylic acid esters and 6-amino-2-2 (heterocyclyl) pyrimidine-4-carboxylic acid esters and their use as herbicides DOW AGROSCIENCES LLC 2015-12-30 CN disclosed
CN-105209452-A 4-amino-6- (heterocyclyl) pyridine-2-carboxylic acid esters and 6-amino-2- (heterocyclyl) pyrimidine-4-carboxylic acid esters and their use as herbicides DOW AGROSCIENCES LLC 2015-12-30 CN disclosed
WO-2015150440-A1 PYRIDINE-2-AMIDES USEFUL AS CB2 AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2015-10-08 WO disclosed
CN-1245401-C 6-aryl-4-aminopicolinates and their use as herbicides DOW AGROSCIENCES LLC (US) 2006-03-15 CN disclosed
CN-1551876-A 6-aryl-4-aminopicolinates and their use as herbicides �ݶ�ũ�����޹�˾ 2004-12-01 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240083908-A1 TETRAHYDROTHIENOPYRIMIDINESULFONAMIDE COMPOUNDS TYMS, TYMP, TPMT NOTUM 1116/4885MAPK1 1982/4885CYP1A2 1688/4885
US-20240368122-A1 JAK2 INHIBITORS AND METHODS OF USE THEREOF JAK2, JAK1, JAK3 NOTUM 2441/4885MAPK1 590/4885CYP1A2 3921/4885
US-20250092033-A1 HETEROAROMATIC NITROGEN-OXIDE COMPOUND, PREPARATION METHOD THEREFOR, AND USE THEREOF CYP19A1, WEE1, WEE2 NOTUM 53/4885MAPK1 3546/4885CYP1A2 130/4885
US-20160340311-A1 RECOVERY AND/OR REUSE OF PALLADIUM CATALYST AFTER A SUZUKI COUPLING DDT, PARK7, DDO NOTUM 1623/4885MAPK1 4248/4885CYP1A2 2325/4885
US-20160376262-A1 NOVEL PYRIDINE DERIVATIVES NDUFS6, NDUFS4, NDUFV1 NOTUM 3969/4885MAPK1 747/4885CYP1A2 60/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.