SCHEMBL17147284

SCHEMBL17147284

Cc1cc(CC(=O)O)cc(C(F)(F)F)c1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RXRA P19793 9/20 0.54
RXRG P48443 9/20 0.54
RXRB P28702 8/20 0.54
AGBL2 Q5U5Z8 1/20 0.49
PSEN1 P49768 1/20 0.46
PSEN2 P49810 1/20 0.46
APH1B Q8WW43 1/20 0.46
NCSTN Q92542 1/20 0.46
APH1A Q96BI3 1/20 0.46
PSENEN Q9NZ42 1/20 0.46
TACR1 P25103 3/20 0.43
PPARG P37231 1/20 0.43
PPARD Q03181 1/20 0.43
PPARA Q07869 1/20 0.43
MRGPRX4 Q96LA9 1/20 0.42
TAS2R14 Q9NYV8 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
FFAR4 Q5NUL3 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29927941 1.00 RXRA (0.54) RXRARXRGRXRBAGBL2PSEN1
SCHEMBL504122 0.87 RXRA (0.68) RXRARXRGRXRBAGBL2PSEN1
SCHEMBL12301741 0.86 TACR1 (0.40) RXRARXRGRXRBAGBL2PSEN1
SCHEMBL22774254 0.84 TACR1 (0.40) RXRARXRGRXRBAGBL2PSEN1
SCHEMBL30875890 0.84 GRIN2B (0.43) RXRARXRGRXRBPSEN1PSEN2
SCHEMBL30151169 0.83 FFAR4 (0.48) RXRARXRGRXRBTACR1PPARA
SCHEMBL29927377 0.83 PSEN1 (0.40) RXRARXRGRXRBAGBL2PSEN1
SCHEMBL22773948 0.82 RXRA (0.54) RXRARXRGRXRBAGBL2PSEN1
SCHEMBL29467110 0.82 RXRA (0.54) RXRARXRGRXRBAGBL2PSEN1
SCHEMBL10137786 0.81 TACR1 (0.41) RXRARXRGRXRBAGBL2PSEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240025895-A1 COMPOSITIONS AND METHODS FOR MODULATING HAIR GROWTH THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2024-01-25 US disclosed
US-11787804-B2 Compositions and methods for modulating hair growth THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-10-17 US disclosed
WO-2022212326-A1 NEK7 INHIBITORS Halia Therapeutics, Inc. (US) 2022-10-06 WO disclosed
US-20220267300-A1 SULFONAMIDE DERIVATIVES AND USES THEREOF NodThera Limited (GB) 2022-08-25 US disclosed
CN-114761383-A Sulfonamide derivatives and uses thereof 诺瑟拉有限公司 2022-07-15 CN disclosed
WO-2020249669-A1 SULFONAMIDE DERIVATIVES AND USES THEREOF NodThera Limited (GB) 2020-12-17 WO disclosed
US-9334249-B2 Inhibitors of cytomegalovirus BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2016-05-10 US disclosed
US-20150284348-A1 INHIBITORS OF CYTOMEGALOVIRUS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-10-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150284348-A1 INHIBITORS OF CYTOMEGALOVIRUS CDKN1A, CCNA1, IFNAR1 RXRA 1227/4885RXRG 2584/4885RXRB 1758/4885
US-20220267300-A1 SULFONAMIDE DERIVATIVES AND USES THEREOF IL1B, IL1A, CASP1 RXRA 2545/4885RXRG 2943/4885RXRB 2384/4885
US-11787804-B2 Compositions and methods for modulating hair growth PC, FH, SLC25A1 RXRA 2175/4885RXRG 1276/4885RXRB 1673/4885
US-20240025895-A1 COMPOSITIONS AND METHODS FOR MODULATING HAIR GROWTH PC, FH, SLC25A1 RXRA 2175/4885RXRG 1276/4885RXRB 1673/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.