SCHEMBL17154

SCHEMBL17154

O=[N+]([O-])c1ccc(S(=O)(=O)Cl)s1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 8/20 0.40
ALDH1A1 P00352 5/20 0.40
MAPT P10636 5/20 0.40
PSMD14 O00487 1/20 0.40
MEN1 O00255 7/20 0.38
CYP2A6 P11509 1/20 0.38
KDM4E B2RXH2 4/20 0.37
L3MBTL1 Q9Y468 4/20 0.37
HTT P42858 2/20 0.37
TDP1 Q9NUW8 1/20 0.37
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA7 P43166 1/20 0.35
CA9 Q16790 1/20 0.35
POLB P06746 3/20 0.35
HSP90AA1 P07900 3/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
LMNA P02545 2/20 0.35
RECQL P46063 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5152682 0.80 MAPT (0.40) KMT2AALDH1A1MAPTPSMD14MEN1
SCHEMBL5227256 0.80 MAPT (0.40) KMT2AALDH1A1MAPTPSMD14MEN1
SCHEMBL1548578 0.80 CA2 (0.44) KMT2AALDH1A1MAPTPSMD14CYP2A6
Hydrochloric Acid SCHEMBL28225407 0.78 MAPT (0.39) KMT2AALDH1A1MAPTPSMD14MEN1
SCHEMBL7132351 0.75 L3MBTL1 (0.46) KMT2AALDH1A1L3MBTL1HTTTDP1
SCHEMBL6261093 0.75 MAPT (0.52) KMT2AALDH1A1MAPTPSMD14MEN1
SCHEMBL10979449 0.73 KMT2A (0.38) KMT2AALDH1A1MAPTMEN1CYP2A6
SCHEMBL5229246 0.72 MEN1 (0.52) KMT2AALDH1A1MAPTMEN1L3MBTL1
SCHEMBL23092462 0.72 GAA (0.39) KMT2AALDH1A1MAPTPSMD14MEN1
SCHEMBL7057572 0.72 APP (0.66) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 45 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105237523-B Pyrimidine derivatives and preparation method thereof, purposes 深圳市博圣康生物科技有限公司 2018-06-01 CN claimed
CN-105237523-A Pyrimidine derivatives, and preparation method and use thereof SHENZHEN BIOSCIEN PHARMACEUTICALS CO LTD 2016-01-13 CN claimed
CN-119899170-A Fluorine-containing thiophene compound, preparation method thereof and electrolyte 江苏华盛锂电材料股份有限公司 2025-04-29 CN disclosed
US-20240262792-A1 USP30 INHIBITORS AND USES THEREOF VINCERE BIOSCIENCES, INC. 2024-08-08 US disclosed
US-11845724-B2 USP30 inhibitors and uses thereof VINCERE BIOSCIENCES, INC. (US) 2023-12-19 US disclosed
US-20230242496-A1 SOX11 INHIBITORS FOR TREATING MANTLE CELL LYMPHOMA ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2023-08-03 US disclosed
EP-4164622-A1 SOX11 INHIBITORS FOR TREATING MANTLE CELL LYMPHOMA Icahn School of Medicine at Mount Sinai (US) 2023-04-19 EP disclosed
US-20220315531-A1 USP30 INHIBITORS AND USES THEREOF VINCERE BIOSCIENCES, INC. 2022-10-06 US disclosed
CN-115038688-A USP30 inhibitors and uses thereof 文森雷生物科学股份有限公司 2022-09-09 CN disclosed
EP-4028385-A1 USP30 INHIBITORS AND USES THEREOF Vincere Biosciences, Inc. (US) 2022-07-20 EP disclosed
WO-2021257544-A1 SOX11 INHIBITORS FOR TREATING MANTLE CELL LYMPHOMA ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2021-12-23 WO disclosed
WO-2004026881-A1 MACROCYCLIC PYRIMIDINES, THE PRODUCTION THEREOF AND THE USE OF THE SAME AS MEDICAMENTS SCHERING AKTIENGESELLSCHAFT (DE) 2004-04-01 WO disclosed
US-20040063737-A1 CDK-inhibitory 2-heteroaryl-pyrimidines, their production and use as pharmaceutical agents SCHERING AG (DE) 2004-04-01 US disclosed
WO-2003076437-A1 CDK INHIBITING 2-HETEROARYL PYRIMIDINE, THE PRODUCTION THEREOF, AND USE THEREOF AS A MEDICAMENT SCHERING AKTIENGESELLSCHAFT (DE) 2003-09-18 WO disclosed
US-6495683-B2 HERPES VIRUS PHARMACIA AND UPJOHN COMPANY 2002-12-17 US disclosed
EP-1159279-B1 4-OXO-4,7-DIHYDRO-THIENO[2,3-B]PYRIDINE-5-CARBOXAMIDES AS ANTIVIRAL AGENTS UPJOHN CO (US) 2002-10-16 EP disclosed
US-20020006937-A1 4-OXO-4,7-dihydro-thieno[2,3-b]pyridine-5-carboxamides as antiviral agents PHARMACIA & UPJOHN COMPANY 2002-01-17 US disclosed
EP-1159279-A2 4-OXO-4,7-DIHYDRO-THIENO[2,3-B]PYRIDINE-5-CARBOXAMIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2001-12-05 EP disclosed
US-6239142-B1 HERPES VIRUS INFECTION PHARMACIA & UPJOHN COMPANY 2001-05-29 US disclosed
WO-2000053610-A2 4-OXO-4,7-DIHYDRO-THIENO[2,3-b]PYRIDINE-5-CARBOXAMIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2000-09-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230242496-A1 SOX11 INHIBITORS FOR TREATING MANTLE CELL LYMPHOMA BCL6, SOX18, BCL3 KMT2A 578/4885ALDH1A1 2654/4885MAPT 4492/4885
US-20040063737-A1 CDK-inhibitory 2-heteroaryl-pyrimidines, their production and use as pharmaceutical agents CDK2, CDK6, CDKL2 KMT2A 634/4885ALDH1A1 2473/4885MAPT 3291/4885
US-20020006937-A1 4-OXO-4,7-dihydro-thieno[2,3-b]pyridine-5-carboxamides as antiviral agents IRF3, IL4, ZC3HAV1 KMT2A 897/4885ALDH1A1 1869/4885MAPT 3930/4885
US-11845724-B2 USP30 inhibitors and uses thereof USP30, USP28, USP1 KMT2A 955/4885ALDH1A1 2021/4885MAPT 2434/4885
US-20220315531-A1 USP30 INHIBITORS AND USES THEREOF USP30, USP28, USP1 KMT2A 955/4885ALDH1A1 2021/4885MAPT 2434/4885
US-20240262792-A1 USP30 INHIBITORS AND USES THEREOF USP30, USP28, USP1 KMT2A 955/4885ALDH1A1 2021/4885MAPT 2434/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.