SCHEMBL172002

SCHEMBL172002

C=C/C(=C\C=C\C(C)(C)C)C(=C)Nc1cccc(-c2c[nH]c(=O)c(N)c2)c1C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 14/20 0.36
AURKA O14965 5/20 0.34
TTK P33981 5/20 0.34
AURKB Q96GD4 5/20 0.34
INCENP Q9NQS7 5/20 0.34
MAPT P10636 2/20 0.34
THRB P10828 2/20 0.34
CASP1 P29466 2/20 0.34
JAK3 P52333 2/20 0.32
BMX P51813 2/20 0.32
TEC P42680 1/20 0.32
TXK P42681 1/20 0.32
ITK Q08881 1/20 0.32
ERBB4 Q15303 1/20 0.32
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
CYP1A2 P05177 1/20 0.31
GLA P06280 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL171447 0.74 BTK (0.54) BTKAURKATTKAURKBINCENP
SCHEMBL171471 0.71 BTK (0.67) BTKBMXITKKDM4EMEN1
SCHEMBL13894283 0.70 BTK (0.53) BTKAURKATTKAURKBINCENP
SCHEMBL13894036 0.67 ITK (0.54) BTKMAPTJAK3BMXITK
SCHEMBL13894035 0.67 TAS1R3 (0.50) AURKATTKAURKBINCENPMAPT
SCHEMBL171444 0.66 BTK (0.45) BTKMAPTJAK3BMXMEN1
SCHEMBL13893955 0.65 DHPS (0.51) BTKALDH1A1LMNA
SCHEMBL13893940 0.63 BTK (0.53) BTKMAPTJAK3BMXKDM4E
SCHEMBL19785758 0.59 KDR (0.43) BTKMAPTKDM4EALDH1A1LMNA
SCHEMBL11448667 0.58 AURKB (0.56) AURKATTKAURKBINCENPMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426109-A1 NOVEL KINASE INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-03-07 EP disclosed