SCHEMBL1729003

SCHEMBL1729003

CNC(=O)CN(CCCN1CCCN(c2nccc(C(F)(F)F)n2)CC1)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.48
HDAC6 Q9UBN7 1/20 0.44
KDM4E B2RXH2 2/20 0.43
HTR1A P08908 4/20 0.42
KMT2A Q03164 1/20 0.42
SLC6A7 Q99884 1/20 0.42
TMEM97 Q5BJF2 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
ADRB1 P08588 1/20 0.39
CHRM4 P08173 1/20 0.39
DRD2 P14416 2/20 0.38
DRD3 P35462 2/20 0.38
CHRM2 P08172 1/20 0.38
CHRM3 P20309 1/20 0.38
ALDH1A1 P00352 1/20 0.37
OPRM1 P35372 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1729313 0.79 PKM (0.55) PKMHDAC6KDM4EHTR1AKMT2A
SCHEMBL3265528 0.79 HDAC6 (0.47) PKMHDAC6KDM4EHTR1AKMT2A
SCHEMBL1729362 0.76 POLB (0.54) PKMKMT2AALDH1A1
SCHEMBL1729007 0.75 PKM (0.47) PKMHDAC6KDM4EHTR1AKMT2A
SCHEMBL1727889 0.73 HTR2A (0.51) HTR1ASIGMAR1DRD2DRD3OPRM1
SCHEMBL1727831 0.72 FAAH (0.47) MAPK1
SCHEMBL1729366 0.72 MAPT (0.47) PKMKDM4EHTR1AKMT2ATMEM97
SCHEMBL9893124 0.72 HDAC6 (0.52) PKMHDAC6KDM4EHTR1ASLC6A7
SCHEMBL16480406 0.71 HDAC6 (0.51) PKMHDAC6KDM4EHTR1ASLC6A7
SCHEMBL3986386 0.71 ADRB1 (0.58) PKMHDAC6KDM4EHTR1AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633735-B1 DERIVATIVES OF PIPERIDINYL- AND PIPERAZINYL-ALKYL CARBAMATES, PREPARATION METHODS THEREOF AND APPLICATION OF SAME IN THERAPEUTICS SANOFI SA (FR) 2011-11-30 EP claimed