SCHEMBL17374754

SCHEMBL17374754

O=C1CCCC2C=C(Oc3ccccc3Cl)C=CC12

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LDHA P00338 3/20 0.36
HPGD P15428 1/20 0.31
KDM4E B2RXH2 1/20 0.30
SLC6A4 P31645 3/20 0.30
SLC6A2 P23975 2/20 0.30
SLC6A3 Q01959 2/20 0.30
CXCL8 P10145 1/20 0.30
CA1 P00915 2/20 0.30
HRH3 Q9Y5N1 1/20 0.30
HTR1A P08908 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7136996 0.74 MRGPRX2 (0.42)
SCHEMBL17374759 0.70
SCHEMBL5483124 0.66
SCHEMBL11512072 0.62 MAOA (0.43) KDM4ESLC6A4SLC6A2SLC6A3CA1
SCHEMBL3293896 0.59 CA1 (0.32) CA1
SCHEMBL1436765 0.59 HPGD (0.59) HPGDSLC6A4SLC6A2SLC6A3CXCL8
SCHEMBL9282009 0.59 LMNA (0.47) LDHAHPGDSLC6A4SLC6A2SLC6A3
SCHEMBL17374755 0.58 LDHA (0.41) LDHAHPGDKDM4ESLC6A4SLC6A2
SCHEMBL21452232 0.58 TP53 (0.44) CA1
SCHEMBL6238119 0.58

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3160952-A1 HISTONE DEMETHYLASE INHIBITORS Celgene Quanticel Research, Inc. (US) 2017-05-03 EP disclosed
WO-2015200709-A1 HISTONE DEMETHYLASE INHIBITORS Quanticel Pharmaceuticals, Inc. (US) 2015-12-30 WO disclosed