SCHEMBL17423697

SCHEMBL17423697

O=C(O)c1c(F)n(F)c2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.47
AGTR1 P30556 8/20 0.45
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 3/20 0.44
HPGD P15428 2/20 0.44
POLB P06746 1/20 0.44
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
GLA P06280 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41
SRC P12931 2/20 0.39
CCR2 P41597 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18614818 0.84 EGFR (0.49) EGFRAGTR1ALDH1A1KDM4EHPGD
SCHEMBL3679414 0.80 AGTR1 (0.51) EGFRAGTR1ALDH1A1KDM4EHPGD
SCHEMBL28246406 0.80 EGFR (0.63) EGFRAGTR1ALDH1A1KDM4EHPGD
SCHEMBL784606 0.76 POLB (0.49) EGFRAGTR1ALDH1A1KDM4EHPGD
SCHEMBL5189056 0.74 KMT2A (0.40) EGFRALDH1A1KDM4EPOLBGLA
SCHEMBL29655556 0.74 KMT2A (0.40) EGFRALDH1A1KDM4EPOLBGLA
SCHEMBL28322929 0.71 AGTR1 (0.50) AGTR1ALDH1A1KDM4EHPGDPOLB
Butyric Acid SCHEMBL9251503 0.70 FABP4 (0.45) EGFRALDH1A1KDM4EHSD17B10
SCHEMBL11959493 0.70 GPR3 (0.55) ALDH1A1KDM4EPOLBMEN1CYP1A2
SCHEMBL9851534 0.69 ATM (0.42) ALDH1A1KDM4EHPGDPOLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3166940-A1 QUINUCLIDINE COMPOUNDS FOR MODULATING ALPHA7 -NICOTINIC ACETYLCHOLINE RECEPTOR ACTIVITY Alpharmagen, LLC (US) 2017-05-17 EP disclosed
WO-2016007630-A1 QUINUCLIDINE COMPOUNDS FOR MODULATING ALPHA7 -NICOTINIC ACETYLCHOLINE RECEPTOR ACTIVITY ALPHARMAGEN, LLC (US) 2016-01-14 WO disclosed