SCHEMBL28322929

SCHEMBL28322929

O=C(O)c1c(-c2ccccc2)c2ccccc2n(F)c1=O

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 3/20 0.50
KMT2A Q03164 2/20 0.50
PADI4 Q9UM07 5/20 0.44
LMNA P02545 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KDM4E B2RXH2 4/20 0.43
RCE1 Q9Y256 1/20 0.43
ALDH1A1 P00352 2/20 0.42
HPGD P15428 2/20 0.42
POLB P06746 2/20 0.42
EDNRB P24530 1/20 0.42
P2RX4 Q99571 1/20 0.41
PTGS2 P35354 1/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5332174 0.78 KMT2A (0.67) KMT2ALMNASMN1; SMN2KDM4ERCE1
SCHEMBL14463630 0.73 PTGS2 (0.58) AGTR1KMT2APADI4LMNASMN1; SMN2
SCHEMBL17423697 0.71 EGFR (0.47) AGTR1KMT2AKDM4EALDH1A1HPGD
SCHEMBL14288833 0.71 ALDH1A1 (0.66) KMT2APADI4LMNASMN1; SMN2KDM4E
SCHEMBL5335958 0.69 TACR1 (0.58) AGTR1KMT2APADI4LMNAKDM4E
SCHEMBL2490336 0.68 AGTR1 (0.53) AGTR1KMT2ALMNASMN1; SMN2KDM4E
SCHEMBL29655556 0.68 KMT2A (0.40) KMT2ALMNAKDM4EALDH1A1POLB
SCHEMBL5189056 0.68 KMT2A (0.40) KMT2ALMNAKDM4EALDH1A1POLB
SCHEMBL29262209 0.68 LMNA (0.55) AGTR1KMT2ALMNAKDM4EALDH1A1
SCHEMBL5339664 0.68 TACR1 (0.59) AGTR1KMT2APADI4LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110248934-A Heteroaryl PAD4 inhibitor 帕德罗科治疗公司 2019-09-17 CN disclosed