SCHEMBL1744740

SCHEMBL1744740

NS(=O)(=O)c1ccccc1-c1ccc(F)cn1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 11/20 0.55
FEN1 P39748 11/20 0.55
PTGS2 P35354 2/20 0.42
PTGS1 P23219 1/20 0.42
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA4 P22748 2/20 0.39
CA6 P23280 2/20 0.39
CA9 Q16790 2/20 0.39
CA12 O43570 1/20 0.39
CYP2C9 P11712 1/20 0.39
CA5A P35218 1/20 0.39
CA7 P43166 1/20 0.39
CA14 Q9ULX7 1/20 0.39
CA5B Q9Y2D0 1/20 0.39
TRPV1 Q8NER1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16180470 0.90 ALOX5AP (0.47) ALOX5APFEN1PTGS2PTGS1CA9
Orthocresol SCHEMBL16180579 0.88 ALOX5AP (0.45) ALOX5APFEN1PTGS2CA1CA2
2-Chlorophenol SCHEMBL16180513 0.88 ALOX5AP (0.45) ALOX5APFEN1PTGS2PTGS1CA1
SCHEMBL16180634 0.87 ALOX5AP (0.47) ALOX5APFEN1
Guaiacol SCHEMBL16180776 0.86 ALOX5AP (0.44) ALOX5APFEN1PTGS2PTGS1CA1
SCHEMBL16180585 0.85 ALOX5AP (0.43) ALOX5APFEN1CA2CA9CA12
SCHEMBL16180522 0.85 ALOX5AP (0.43) ALOX5APFEN1PTGS2CA9
SCHEMBL31234503 0.83 ALOX5AP (0.43) ALOX5APFEN1PTGS2PTGS1CA2
SCHEMBL16177988 0.81 PTGS2 (0.50) ALOX5APFEN1PTGS2CA1CA2
SCHEMBL6883474 0.80 KIF11 (0.50) ALOX5APFEN1TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4716529-A2 COMPOUNDS THAT RE-ACTIVATE MUTANT P53 Institute For Cancer Research d/b/a The Research Institute of Fox Chase Cancer Center (US) 2026-04-01 EP disclosed
WO-2024243343-A2 COMPOUNDS THAT RE-ACTIVATE MUTANT P53 KARANICOLAS JOHN (US) 2024-11-28 WO disclosed
US-20150259327-A1 Chemical Compounds PFIZER LIMITED (GB) 2015-09-17 US disclosed
US-9067922-B2 Chemical compounds PFIZER LIMITED (GB) 2015-06-30 US disclosed
US-8907101-B2 Sulfonamide derivatives PFIZER LIMITED (GB) 2014-12-09 US disclosed
US-20140315878-A1 CHEMICAL COMPOUNDS PFIZER LIMITED (GB) 2014-10-23 US disclosed
US-20130338111-A1 Sulfonamide Derivatives ICAGEN, INC. (US) 2013-12-19 US disclosed
US-20120149679-A1 Sulfonamide Derivatives ICAGEN, INC. 2012-06-14 US disclosed
EP-2385938-A1 SULFONAMIDE DERIVATIVES Pfizer Limited (GB) 2011-11-16 EP disclosed
US-8040476-B2 Display device and method of producing the same MITSUBISHI ELECTRIC CORPORATION (JP) 2011-10-18 US disclosed
US-20100197655-A1 SULFONAMIDE DERIVATIVES Pfizer Limited Icagen, Inc. 2010-08-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100197655-A1 SULFONAMIDE DERIVATIVES SULT2A1, SULT1A1, TPST2 ALOX5AP 1186/4885FEN1 4863/4885PTGS2 209/4885
US-20130338111-A1 Sulfonamide Derivatives SULT2A1, SULT1A1, TPST2 ALOX5AP 1186/4885FEN1 4863/4885PTGS2 209/4885
US-20150259327-A1 Chemical Compounds SULT2A1, SULT1A1, SULT1E1 ALOX5AP 4059/4885FEN1 4600/4885PTGS2 3678/4885
US-20140315878-A1 CHEMICAL COMPOUNDS SULT2A1, SULT1A1, SULT1E1 ALOX5AP 4059/4885FEN1 4600/4885PTGS2 3678/4885
US-20120149679-A1 Sulfonamide Derivatives SULT2A1, SULT1A1, TPST2 ALOX5AP 1186/4885FEN1 4863/4885PTGS2 209/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.