SCHEMBL17469288

SCHEMBL17469288

COc1cc2c(C(=O)C(F)(F)F)c(C(F)(F)F)n(C)c2cc1-c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
RET P07949 1/20 0.40
BACE1 P56817 1/20 0.39
KDM4E B2RXH2 2/20 0.38
ATM Q13315 1/20 0.37
ALDH1A1 P00352 5/20 0.37
LDHA P00338 1/20 0.36
AKR1C3 P42330 2/20 0.36
AKR1C2 P52895 2/20 0.36
IDO1 P14902 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
MLYCD O95822 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17469291 0.82 KMT2A (0.56) MEN1KMT2AL3MBTL1ALDH1A1IDO1
SCHEMBL17469290 0.81 KMT2A (0.42) MEN1KMT2AL3MBTL1KDM4EATM
SCHEMBL17469277 0.81 KMT2A (0.40) MEN1KMT2AL3MBTL1ATMALDH1A1
SCHEMBL17469283 0.80 MEN1 (0.39) MEN1KMT2AL3MBTL1ALDH1A1LMNA
SCHEMBL17469287 0.80 KMT2A (0.39) MEN1KMT2AL3MBTL1ATMALDH1A1
SCHEMBL17469272 0.75 MAPT (0.45) MEN1KMT2AL3MBTL1KDM4EALDH1A1
SCHEMBL19322245 0.74 KDM4E (0.40) MEN1KMT2ABACE1KDM4EATM
SCHEMBL24236617 0.71 TSHR (0.45) KDM4EALDH1A1MAPT
SCHEMBL24236616 0.66 PLA2G2A (0.58) MEN1KMT2AALDH1A1
SCHEMBL28032229 0.66 TUBB4A (0.41) MEN1KMT2AKDM4EALDH1A1S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016014426-A1 ORGANIC REACTIONS THE ARIZONA BOARD OF REGENTS (US) 2016-01-28 WO disclosed