SCHEMBL17469283

SCHEMBL17469283

COc1cc2c(C(=O)C(F)(F)F)c(C(F)(F)F)n(C)c2cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
RORC P51449 3/20 0.36
ALDH1A1 P00352 1/20 0.36
KMO O15229 1/20 0.36
LMNA P02545 3/20 0.35
TSHR P16473 1/20 0.35
CYP1A1 P04798 1/20 0.35
CYP1B1 Q16678 1/20 0.35
TP53 P04637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
BCAT2 O15382 1/20 0.34
BCAT1 P54687 1/20 0.34
MTNR1A P48039 1/20 0.34
MTNR1B P49286 1/20 0.34
PLA2G2A P14555 1/20 0.34
S1PR2 O95136 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17469290 0.86 KMT2A (0.42) MEN1KMT2AL3MBTL1RORCALDH1A1
SCHEMBL17469277 0.86 KMT2A (0.40) MEN1KMT2AL3MBTL1RORCALDH1A1
SCHEMBL17469287 0.85 KMT2A (0.39) MEN1KMT2AL3MBTL1RORCALDH1A1
SCHEMBL17469291 0.85 KMT2A (0.56) MEN1KMT2AL3MBTL1ALDH1A1LMNA
SCHEMBL17469288 0.80 MEN1 (0.40) MEN1KMT2AL3MBTL1ALDH1A1LMNA
SCHEMBL17469272 0.77 MAPT (0.45) MEN1KMT2AL3MBTL1ALDH1A1NPSR1
SCHEMBL19322240 0.71 MTNR1A (0.42) MEN1KMT2AL3MBTL1ALDH1A1LMNA
SCHEMBL24236617 0.69 TSHR (0.45) ALDH1A1TSHRMTNR1AMTNR1BPLA2G2A
SCHEMBL17469273 0.66 POLB (0.46) ALDH1A1LMNATSHRNPSR1MTNR1A
SCHEMBL17469278 0.66 KDM4E (0.44) MEN1KMT2AALDH1A1LMNAMTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016014426-A1 ORGANIC REACTIONS THE ARIZONA BOARD OF REGENTS (US) 2016-01-28 WO disclosed