SCHEMBL17524933

SCHEMBL17524933

COc1cc(N2CCC3(CC2)C(=O)Nc2ncccc23)ccc1N

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CALCA P06881 3/20 0.40
MALT1 Q9UDY8 1/20 0.39
MAP3K11 Q16584 1/20 0.39
CHEK1 O14757 1/20 0.39
CALCRL Q16602 2/20 0.37
PLD2 O14939 1/20 0.37
PLD1 Q13393 1/20 0.37
EGLN1 Q9GZT9 2/20 0.36
JAK2 O60674 2/20 0.36
JAK1 P23458 1/20 0.36
TYK2 P29597 1/20 0.36
JAK3 P52333 1/20 0.36
IDH1 O75874 2/20 0.35
ALK Q9UM73 1/20 0.35
AVPR1A P37288 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
DPP4 P27487 1/20 0.35
HTR1A P08908 1/20 0.35
HTR2A P28223 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17524942 0.90 ADRA2B (0.40) CALCACALCRLEGLN1IDH1ALDH1A1
SCHEMBL17524907 0.90 MALT1 (0.41) CALCAMALT1MAP3K11CALCRLEGLN1
SCHEMBL17524873 0.87 HTR6 (0.38) CALCACALCRLEGLN1HTR1AHTR2A
SCHEMBL17524935 0.86 GAA (0.44) CALCAMALT1CALCRLEGLN1HTR1A
SCHEMBL17524946 0.85 CALCRL (0.38) CALCACALCRLIDH1ALDH1A1HTR1A
SCHEMBL17524957 0.85 CALCA (0.38) CALCACALCRLIDH1HTR1AHTR2A
SCHEMBL17524951 0.85 LTA4H (0.38) CALCACALCRLHTR1AHTR2AHTR7
SCHEMBL17524940 0.84 CALCA (0.40) CALCACALCRLHTR1AHTR2AHTR7
SCHEMBL17524938 0.84 HTR7 (0.45) CALCAMALT1CALCRLLMNAHTR1A
SCHEMBL17524901 0.82 ADRA2B (0.40) CALCAMALT1CALCRLEGLN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016022644-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-02-11 WO disclosed