SCHEMBL17524938

SCHEMBL17524938

Nc1ccc(N2CCC3(CC2)C(=O)Nc2ncccc23)cc1Cl

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 9/20 0.45
HTR1A P08908 6/20 0.45
HTR2A P28223 6/20 0.45
HTR6 P50406 6/20 0.45
CALCA P06881 4/20 0.40
MALT1 Q9UDY8 1/20 0.37
CALCRL Q16602 4/20 0.36
MMP2 P08253 1/20 0.35
MMP13 P45452 1/20 0.35
ADAM17 P78536 1/20 0.35
ADAMTS1 Q9UHI8 1/20 0.35
ADAMTS5 Q9UNA0 1/20 0.35
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
ALOX12 P18054 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17525077 0.89 HTR7 (0.46) HTR7HTR1AHTR2AHTR6CALCA
SCHEMBL17524935 0.87 GAA (0.44) HTR7HTR1AHTR2AHTR6CALCA
SCHEMBL17524940 0.87 CALCA (0.40) HTR7HTR1AHTR2AHTR6CALCA
SCHEMBL17524933 0.84 CALCA (0.40) HTR7HTR1AHTR2AHTR6CALCA
SCHEMBL17524923 0.83 CALCA (0.41) HTR7HTR1AHTR2AHTR6CALCA
SCHEMBL17524942 0.82 ADRA2B (0.40) HTR7HTR1AHTR2AHTR6CALCA
SCHEMBL17524910 0.82 EGLN1 (0.43) HTR7HTR1AHTR2AHTR6CALCA
SCHEMBL17524873 0.81 HTR6 (0.38) HTR7HTR1AHTR2AHTR6CALCA
SCHEMBL17525019 0.80 MAPK1 (0.41) HTR7HTR1AHTR2AHTR6CALCA
SCHEMBL17524957 0.80 CALCA (0.38) HTR7HTR1AHTR2AHTR6CALCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016022644-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-02-11 WO disclosed