SCHEMBL175502

SCHEMBL175502

Nc1nc(-c2ccccc2)c(C(=O)c2ccc3c(c2)OCO3)s1

nearest known ligand 0.61

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CFTR P13569 18/20 0.61
HPGD P15428 1/20 0.49
RAB9A P51151 1/20 0.49
LIMK1 P53667 1/20 0.49
TP53 P04637 1/20 0.48
MAPT P10636 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14264462 0.81 RAB9A (0.49) CFTRHPGDRAB9ALIMK1TP53
SCHEMBL165773 0.79 ADORA3 (0.61) MAPT
SCHEMBL27653923 0.78 ALDH1A1 (0.64) MAPT
SCHEMBL4880488 0.78 FBP1 (0.57)
SCHEMBL257616 0.76 ADORA3 (0.64) HPGDRAB9AMAPT
SCHEMBL10092883 0.76 RORB (0.67)
SCHEMBL18411276 0.75 CDK4 (0.55) HPGDRAB9ALIMK1TP53MAPT
SCHEMBL2762916 0.72 ALDH1A1 (0.64) MAPT
SCHEMBL7816239 0.72 SRD5A2 (0.81) HPGDRAB9AMAPT
SCHEMBL976273 0.71 CDC7 (0.60) CFTRHPGDRAB9ATP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012027965-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-08 WO disclosed
WO-2012027965-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-08 WO disclosed