SCHEMBL17844206

SCHEMBL17844206

Cc1cc(CNc2c(-c3ccccc3)sn(C(C)(C)C)c2=O)no1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
GRIN1 Q05586 3/20 0.39
GRIN2B Q13224 3/20 0.39
MAPT P10636 1/20 0.39
RECQL P46063 1/20 0.39
GABRA5 P31644 2/20 0.36
BRAF P15056 1/20 0.36
GABRA1 P14867 1/20 0.35
FEN1 P39748 1/20 0.34
HTR2A P28223 1/20 0.34
KCNH2 Q12809 1/20 0.34
TLR7 Q9NYK1 1/20 0.34
SYK P43405 1/20 0.34
GPR142 Q7Z601 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
EPHX2 P34913 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20678598 0.80 GABRA5 (0.49) MAPTGABRA5
SCHEMBL17844243 0.80 PRKAA2 (0.43) GRIN1GRIN2BMAPTRECQLGABRA5
SCHEMBL3551960 0.79 BRD4 (0.39) MAPTRECQL
SCHEMBL5184298 0.72 CA12 (0.33) MAPTKCNH2
SCHEMBL17844229 0.72 MEN1 (0.48) NPC1RAB9AMAPTRECQLMAPK1
SCHEMBL17844110 0.72 MAOA (0.40)
SCHEMBL17844227 0.71 POLB (0.39) MAPTSYKMAPK1
SCHEMBL17844175 0.71 CA12 (0.38) MAPTCYP2C19
SCHEMBL17844228 0.71 CYP1A2 (0.43) MAPTGABRA5GABRA1CYP1A2CYP2D6
SCHEMBL3653144 0.70 SMN1; SMN2 (0.36) KCNH2SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016100619-A2 TREATMENT AND DIAGNOSIS OF CANCER RGENIX, INC. (US) 2016-06-23 WO disclosed