SCHEMBL17850360

SCHEMBL17850360

O=C(NCc1c(F)ccc(F)c1Cl)C1=C(C2CC2)NNS1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 13/20 0.43
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
MET P08581 2/20 0.38
FPR3 P25089 1/20 0.35
ATM Q13315 1/20 0.33
ALDH2 P05091 1/20 0.32
INPPL1 O15357 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17850365 0.84 ATM (0.46) P2RX7ROCK2ROCK1METATM
SCHEMBL17850362 0.84 P2RX7 (0.39) P2RX7ATM
SCHEMBL17850355 0.84 ATM (0.45) P2RX7ROCK2ROCK1METATM
SCHEMBL17850366 0.84 ATM (0.45) P2RX7ROCK2ROCK1METATM
SCHEMBL17850367 0.79 P2RX7 (0.45) P2RX7ROCK2ROCK1ATM
SCHEMBL17850358 0.75 LMNA (0.58) ATM
SCHEMBL13938088 0.71 ATM (0.51) P2RX7ROCK2ROCK1METFPR3
SCHEMBL4598761 0.70 P2RX7 (0.60) P2RX7FPR3
SCHEMBL17850357 0.68 ATM (0.56) P2RX7ROCK2ROCK1METATM
SCHEMBL17850363 0.68 MAPK14 (0.44) P2RX7ROCK2ROCK1ATMINPPL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3034494-A1 HETEROCYCLIC INHIBITORS OF NECROPTOSIS President and Fellows of Harvard College (US) 2016-06-22 EP disclosed