SCHEMBL17850362

SCHEMBL17850362

O=C(NCc1c(Cl)cccc1Cl)C1=C(C2CC2)NNS1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 11/20 0.39
KMT2A Q03164 1/20 0.39
LMNA P02545 1/20 0.38
GLA P06280 1/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ATM Q13315 1/20 0.37
POLB P06746 1/20 0.35
SLC6A3 Q01959 1/20 0.35
MAPK1 P28482 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17850367 0.93 P2RX7 (0.45) P2RX7LMNAATMMAPK1
SCHEMBL17850365 0.90 ATM (0.46) P2RX7KMT2AATMPOLBCYP1A2
SCHEMBL17850366 0.89 ATM (0.45) P2RX7KMT2AATM
SCHEMBL17850355 0.89 ATM (0.45) P2RX7KMT2AATMPOLBCYP1A2
SCHEMBL17850358 0.89 LMNA (0.58) KMT2ALMNAHTTNPSR1ATM
SCHEMBL17850360 0.84 P2RX7 (0.43) P2RX7ATM
SCHEMBL17850357 0.73 ATM (0.56) P2RX7LMNAATMPOLB
SCHEMBL12852318 0.68 ATM (0.58) P2RX7KMT2ALMNAHTTATM
SCHEMBL17850363 0.65 MAPK14 (0.44) P2RX7KMT2AATM
SCHEMBL13938748 0.65 SLC6A3 (0.35) LMNASLC6A3MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3034494-A1 HETEROCYCLIC INHIBITORS OF NECROPTOSIS President and Fellows of Harvard College (US) 2016-06-22 EP disclosed