SCHEMBL17850367

SCHEMBL17850367

Cc1cccc(Cl)c1CNC(=O)C1=C(C2CC2)NNS1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 14/20 0.45
DGAT1 O75907 1/20 0.42
MAPK1 P28482 1/20 0.38
ATM Q13315 1/20 0.38
LMNA P02545 1/20 0.37
ROCK2 O75116 1/20 0.36
ROCK1 Q13464 1/20 0.36
HDAC8 Q9BY41 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17850362 0.93 P2RX7 (0.39) P2RX7MAPK1ATMLMNA
SCHEMBL17850365 0.84 ATM (0.46) P2RX7ATMROCK2ROCK1
SCHEMBL17850355 0.83 ATM (0.45) P2RX7ATMROCK2ROCK1
SCHEMBL17850366 0.83 ATM (0.45) P2RX7ATMROCK2ROCK1
SCHEMBL17850358 0.83 LMNA (0.58) ATMLMNA
SCHEMBL17850360 0.79 P2RX7 (0.43) P2RX7ATMROCK2ROCK1
SCHEMBL17850357 0.73 ATM (0.56) P2RX7ATMLMNAROCK2ROCK1
SCHEMBL12852300 0.72 ATM (0.57) P2RX7DGAT1MAPK1ATM
SCHEMBL5798009 0.67 P2RX7 (0.54) P2RX7MAPK1LMNAHDAC8
SCHEMBL17850363 0.65 MAPK14 (0.44) P2RX7ATMROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3034494-A1 HETEROCYCLIC INHIBITORS OF NECROPTOSIS President and Fellows of Harvard College (US) 2016-06-22 EP disclosed