SCHEMBL17899709

SCHEMBL17899709

CN1CCN(c2ccc(-c3ccc(S(=O)(=O)Cl)cc3)cc2)CC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.50
MEN1 O00255 1/20 0.50
HTT P42858 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
CHKA P35790 1/20 0.50
SIRT6 Q8N6T7 1/20 0.50
MAP4K1 Q92918 1/20 0.49
CHEK1 O14757 1/20 0.49
ALDH1A1 P00352 3/20 0.49
KDM4E B2RXH2 2/20 0.49
MAPT P10636 2/20 0.49
GAA P10253 1/20 0.49
ADRA2C P18825 1/20 0.49
GFER P55789 1/20 0.49
PTK2B Q14289 1/20 0.49
ESR2 Q92731 1/20 0.49
JAK2 O60674 2/20 0.48
JAK3 P52333 1/20 0.48
PTK2 Q05397 1/20 0.48
LSS P48449 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17897423 0.85 HTR2C (0.49) ALDH1A1ADRA2CJAK2JAK3PTK2
SCHEMBL7652825 0.84 LMNA (0.54) HTTCHKAALDH1A1KDM4EMAPT
SCHEMBL7652722 0.83 LMNA (0.53) KMT2AMEN1HTTL3MBTL1ALDH1A1
SCHEMBL17902923 0.83 KDM4E (0.53) KMT2ACHKAALDH1A1KDM4EMAPT
SCHEMBL17902922 0.82 RPS6KA3 (0.45) KMT2ACHKASIRT6GFERJAK2
SCHEMBL6561315 0.81 PKM (0.58) KMT2AMEN1HTTALDH1A1KDM4E
SCHEMBL17897410 0.80 MEN1 (0.37) KMT2AMEN1HTTL3MBTL1MAP4K1
SCHEMBL17902921 0.80 ALDH1A1 (0.63) HTTSIRT6ALDH1A1KDM4ETSHR
SCHEMBL28170767 0.79 AKR1C3 (0.58) KMT2AMEN1SIRT6MAP4K1ALDH1A1
SCHEMBL6877901 0.79 SIRT6 (0.56) KMT2AMEN1CHKASIRT6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016107542-A1 PYRROLE AMIDE COMPOUND, PREPARATION METHOD THEREFOR, AND USE THEREOF 成都先导药物开发有限公司 2016-07-07 WO disclosed
WO-2016107544-A1 INTERMEDIATE COMPOUND FOR PREPARING PYRROLE AMIDE COMPOUND AND PREPARATION METHOD AND USE THEREOF 成都先导药物开发有限公司 2016-07-07 WO disclosed
CN-105732458-A Pyrrole amide compounds, preparation method and applications thereof 成都先导药物开发有限公司 2016-07-06 CN disclosed