SCHEMBL18061111

SCHEMBL18061111

CC(C(=O)O)c1cccc(-c2ccccc2)c1NC(=O)Nc1ccncc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.51
ALDH1A1 P00352 2/20 0.49
MDM2 Q00987 1/20 0.45
SMN1; SMN2 Q16637 3/20 0.44
KMT2A Q03164 3/20 0.44
PKM P14618 1/20 0.44
POLB P06746 2/20 0.42
LMNA P02545 1/20 0.42
STAT3 P40763 1/20 0.42
EGFR P00533 1/20 0.42
FGFR1 P11362 1/20 0.42
KDR P35968 1/20 0.42
CCKBR P32239 1/20 0.41
MEN1 O00255 1/20 0.41
ROCK2 O75116 3/20 0.41
CYP3A4 P08684 1/20 0.41
CYP3A5 P20815 1/20 0.41
ROCK1 Q13464 2/20 0.40
CNR1 P21554 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL339362 0.79 CXCL8 (0.46) ALDH1A1SMN1; SMN2KMT2APOLBLMNA
SCHEMBL341017 0.78 KMT2A (0.45) ALDH1A1SMN1; SMN2KMT2APOLBLMNA
SCHEMBL5642336 0.76 MDM2 (0.59) TAAR1ALDH1A1MDM2SMN1; SMN2KMT2A
SCHEMBL338541 0.76 MAPT (0.43) ALDH1A1SMN1; SMN2KMT2APOLBMEN1
SCHEMBL341491 0.74 SOAT1 (0.46) ALDH1A1SMN1; SMN2KMT2ALMNAMEN1
SCHEMBL18061112 0.74 TAAR1 (0.51) TAAR1ALDH1A1MDM2SMN1; SMN2KMT2A
SCHEMBL341352 0.72 LMNA (0.50) ALDH1A1MDM2SMN1; SMN2KMT2APOLB
SCHEMBL2393839 0.71 PTGS2 (0.56) SMN1; SMN2KMT2ALMNAMEN1
SCHEMBL305498 0.71 TAAR1 (1.00) TAAR1ALDH1A1MDM2SMN1; SMN2KMT2A
Biphenyl SCHEMBL7876282 0.70 PTGS2 (0.58) KMT2APKMLMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2776389-B1 ARYL UREA DERIVATIVES AS N-FORMYL PEPTIDE RECEPTOR LIKE-1 (FPRL-1) RECEPTOR MODULATORS ALLERGAN INC (US) 2016-09-21 EP claimed