SCHEMBL1809848

SCHEMBL1809848

O=[N+]([O-])c1nc(Br)ccc1O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.37
TP53 P04637 2/20 0.37
HPGD P15428 2/20 0.37
TSHR P16473 2/20 0.37
MAPK1 P28482 2/20 0.37
ALDH1A1 P00352 2/20 0.37
GPR35 Q9HC97 1/20 0.37
CTSB P07858 4/20 0.37
CTSH P09668 1/20 0.37
MAPT P10636 3/20 0.36
HTT P42858 2/20 0.36
POLB P06746 1/20 0.36
GAA P10253 2/20 0.36
CYP3A4 P08684 1/20 0.36
HIF1A Q16665 1/20 0.36
THRB P10828 1/20 0.36
ALOX15 P16050 1/20 0.36
HSD17B10 Q99714 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TDP1 Q9NUW8 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30152695 1.00 SMN1; SMN2 (0.37) SMN1; SMN2TP53HPGDTSHRMAPK1
SCHEMBL3827420 0.87 MAPT (0.43) SMN1; SMN2TSHRALDH1A1CTSBMAPT
SCHEMBL19122111 0.82
SCHEMBL3829294 0.80 MAPT (0.44) SMN1; SMN2MAPK1ALDH1A1MAPTHTT
SCHEMBL3829304 0.80 MAPT (0.44) SMN1; SMN2MAPK1ALDH1A1MAPTHTT
SCHEMBL19135896 0.80 SMN1; SMN2 (0.37) SMN1; SMN2TP53HPGDTSHRMAPK1
SCHEMBL18979820 0.79 MAPT (0.37) SMN1; SMN2HPGDMAPK1ALDH1A1MAPT
SCHEMBL30370409 0.79 MAPT (0.37) SMN1; SMN2HPGDMAPK1ALDH1A1MAPT
SCHEMBL23041103 0.78 ALDH1A1 (0.50) SMN1; SMN2TP53HPGDTSHRMAPK1
SCHEMBL29769754 0.78 ALDH1A1 (0.50) SMN1; SMN2TP53HPGDTSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 373 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102977117-A Method for synthesizing 6-bromo-2, 2-dimethyl-2H-pyridino [3, 2-B] [1, 4] oxazine-3(4H)-one CGENE TECH SUZHOU CHINA CO LTD 2013-03-20 CN claimed
US-20260035362-A1 GLP-1R AGONISTS AND USES THEREOF QILU REGOR THERAPEUTICS INC (CN) 2026-02-05 US disclosed
EP-4608831-A1 COMPOUNDS AND USES THEREOF Suzhou Zanrong Pharma Limited (CN) 2025-09-03 EP disclosed
US-12365670-B2 GLP-IR agonists and uses thereof QILU REGOR THERAPEUTICS INC. (CN) 2025-07-22 US disclosed
US-20250205232-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2025-06-26 US disclosed
US-20250163038-A1 CBL-B MODULATORS AND USES THEREOF NIMBUS CLIO, INC. 2025-05-22 US disclosed
CN-119431398-A Anti-tumor application of R406 and derivatives thereof in cooperation with TRAIL 中国科学院上海有机化学研究所 2025-02-14 CN disclosed
WO-2024259241-A1 5-HT2A RECEPTOR MODULATORS AND METHODS OF USE THEREOF Transneural Therapeutics, Inc. (US) 2024-12-19 WO disclosed
US-12168009-B2 Modulators of cystic fibrosis transmembrane conductance regulator VERTEX PHARMACEUTICALS INCORPORATED (US) 2024-12-17 US disclosed
US-20240368189-A1 Modulators of Cystic Fibrosis Transmembrane Conductance Regulator, Pharmaceutical Compositions, Methods of Treatment, and Process for Making the Modulators VERTEX PHARMA (US) 2024-11-07 US disclosed
EP-1549156-A1 DENATURED CAROB FLOUR (DCF) WITH A LOW CONTENT OF SOLUBLE TANNINS AND SUGARS, MEANT FOR HUMAN CONSUMPTION AND PROCESS TO OBTAIN IT Investigacion Y Nutricion, S.L. (ES) 2005-07-06 EP disclosed
EP-1470125-A1 AMINOPIPERIDINE DERIVATIVES GLAXO GROUP LIMITED (GB) 2004-10-27 EP disclosed
CN-1535272-A Nitrogen-containing bicyclic heterocycles ʷ 2004-10-06 CN disclosed
US-20040171620-A1 Nitrogen-containing bicyclic heterocycles for use as antibacterials SMITHKLINE BEECHAM P.L.C. (GB) 2004-09-02 US disclosed
WO-2004058144-A2 ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2004-07-15 WO disclosed
US-20040138219-A1 Quinolines and nitrogenated derivative therof substituted in 4-position by a piperidine-containing moiety and their use as antibacterial agents SMITHKLINE BEECHAM P.L.C. (GB) 2004-07-15 US disclosed
WO-2004014361-A9 AMINOCYCLOHEXENE QUINOLINES AND THEIR AZAISOSTERIC ANALOGUES WITH ANTIBACTERIAL ACTIVITY GLAXO GROUP LTD (GB) 2004-04-08 WO disclosed
WO-2004014150-A1 DENATURED CAROB FLOUR (DCF) WITH A LOW CONTENT OF SOLUBLE TANNINS AND SUGARS, MEANT FOR HUMAN CONSUMPTION AND PROCESS TO OBTAIN IT INVESTIGACION Y NUTRICION, S.L. (ES) 2004-02-19 WO disclosed
WO-2004002490-A2 PIPERIDINE COMPOUNDS AS ANTIBACTERIALS GLAXO GROUP LIMITED (GB) 2004-01-08 WO disclosed
WO-2003064421-A1 AMINOPIPERIDINE DERIVATIVES GLAXO GROUP LIMITED (GB) 2003-08-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260035362-A1 GLP-1R AGONISTS AND USES THEREOF GLP1R, GPR119, IAPP SMN1; SMN2 1240/4885TP53 4567/4885HPGD 3538/4885
US-20040171620-A1 Nitrogen-containing bicyclic heterocycles for use as antibacterials NRDC, NUCB2, NDC1 SMN1; SMN2 1588/4885TP53 3059/4885HPGD 58/4885
US-20250163038-A1 CBL-B MODULATORS AND USES THEREOF CBLB, CBL, CBLC SMN1; SMN2 3005/4885TP53 378/4885HPGD 4374/4885
US-12365670-B2 GLP-IR agonists and uses thereof GLP1R, GPR119, GIPR SMN1; SMN2 3874/4885TP53 4880/4885HPGD 1510/4885
US-20250205232-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR CFTR, SCNN1B, SLC26A4 SMN1; SMN2 4751/4885TP53 4503/4885HPGD 1850/4885
US-20240368189-A1 Modulators of Cystic Fibrosis Transmembrane Conductance Regulator, Pharmaceutical Compositions, Methods of Treatment, and Process for Making the Modulators CFTR, SLC26A4, ABCB11 SMN1; SMN2 4761/4885TP53 4508/4885HPGD 144/4885
US-20040138219-A1 Quinolines and nitrogenated derivative therof substituted in 4-position by a piperidine-containing moiety and their use as antibacterial agents NCF1, TEAD1, TYMS SMN1; SMN2 2305/4885TP53 1717/4885HPGD 746/4885
US-12168009-B2 Modulators of cystic fibrosis transmembrane conductance regulator CFTR, SCNN1B, SLC26A4 SMN1; SMN2 4751/4885TP53 4503/4885HPGD 1850/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.