SCHEMBL18153950

SCHEMBL18153950

O=C(O)c1ccc2c(c1)CC(C1CCCCC1)C1(CCNCC1)O2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.41
RXRA P19793 2/20 0.37
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRM1 P35372 1/20 0.34
KDM1A O60341 2/20 0.34
ALDH1A1 P00352 3/20 0.33
KMO O15229 1/20 0.33
MAPK1 P28482 1/20 0.33
PGR P06401 1/20 0.32
NR3C2 P08235 1/20 0.32
NPC1 O15118 3/20 0.32
RAB9A P51151 3/20 0.32
TP53 P04637 1/20 0.32
HPGD P15428 1/20 0.32
NFKB1 P19838 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18145102 0.71 OPRM1 (0.39) TDP1OPRD1OPRM1KDM1ASMYD3
SCHEMBL3837866 0.67 OPRD1 (0.42) TDP1RXRAOPRD1OPRM1ALDH1A1
SCHEMBL3836335 0.66 OPRD1 (0.36) TDP1RXRAOPRD1ALDH1A1MAPK1
Hydrochloric Acid SCHEMBL1814403 0.64 OPRD1 (0.36) TDP1RXRAOPRD1
SCHEMBL18153948 0.64 HRH3 (0.57)
SCHEMBL2175673 0.63 RXRA (0.56) TDP1RXRAKDM4EMAPTKDM1A
Piperidine SCHEMBL11861125 0.63 KDM4E (0.42) TDP1RXRAKDM4EMAPTALDH1A1
SCHEMBL30948434 0.62 ALDH1A1 (0.46) TDP1RXRAKDM4EMAPTKDM1A
SCHEMBL30948433 0.62 ALDH1A1 (0.46) TDP1RXRAKDM4EMAPTKDM1A
SCHEMBL743920 0.61 HDAC3 (0.61) KDM4EOPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016168660-A1 3-SPIRO-7-HYDROXAMIC ACID TETRALINS AS HDAC INHIBITORS FORMA THERAPEUTICS, INC. (US) 2016-10-20 WO disclosed