SCHEMBL18166321

SCHEMBL18166321

Cc1ccc(-c2cc(OC(=O)NC(C)c3cccnc3)cc(-n3cnnn3)c2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.44
P2RX3 P56373 3/20 0.39
P2RX2 Q9UBL9 3/20 0.39
CTSK P43235 1/20 0.38
TSHR P16473 1/20 0.38
PTGS2 P35354 1/20 0.37
ROCK1 Q13464 5/20 0.36
PRKG1 Q13976 3/20 0.36
CHEK1 O14757 2/20 0.36
RPS6KA5 O75582 2/20 0.36
PRKCG P05129 2/20 0.36
CDK1 P06493 2/20 0.36
PRKACA P17612 2/20 0.36
RPS6KB1 P23443 2/20 0.36
CDK2 P24941 2/20 0.36
MAPK1 P28482 2/20 0.36
AKT2 P31751 2/20 0.36
GSK3A P49840 2/20 0.36
GSK3B P49841 2/20 0.36
IRAK1 P51617 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18166313 0.90 KMT2A (0.42) KMT2AP2RX3P2RX2CTSKTSHR
SCHEMBL18166425 0.90 KMT2A (0.44) KMT2AP2RX3P2RX2CTSKTSHR
SCHEMBL18166303 0.88 ROCK1 (0.39) KMT2AP2RX3P2RX2CTSKTSHR
SCHEMBL18166305 0.87 P2RX3 (0.53) P2RX3P2RX2
SCHEMBL18166309 0.86 KMT2A (0.46) KMT2AP2RX3P2RX2CTSKTSHR
SCHEMBL10243012 0.86 P2RX3 (0.51) P2RX3P2RX2TSHRROCK1PRKG1
SCHEMBL18166377 0.84 KMT2A (0.44) KMT2AP2RX3P2RX2TSHRTP53
SCHEMBL18166327 0.84 ROCK1 (0.39) CTSKTSHRPTGS2ROCK1PRKG1
SCHEMBL18166408 0.84 MARS1 (0.46) KMT2AROCK1ROCK2DGAT2
SCHEMBL18166395 0.83 KMT2A (0.41) KMT2AP2RX3P2RX2TSHRTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2038264-B1 TETRAZOLE-SUBSTITUTED ARYLAMIDES HOFFMANN LA ROCHE (CH) 2016-10-26 EP claimed