SCHEMBL1853274

SCHEMBL1853274

CS(=O)(=O)c1ccc(CCC(N)=O)nc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.42
ALDH1A1 P00352 2/20 0.42
MBOAT4 Q96T53 1/20 0.40
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
KCNH2 Q12809 1/20 0.39
PRMT1 Q99873 1/20 0.37
MAP4K4 O95819 1/20 0.36
JAK2 O60674 1/20 0.36
FFAR1 O14842 1/20 0.36
GSR P00390 1/20 0.36
LOX P28300 1/20 0.35
LOXL2 Q9Y4K0 1/20 0.35
NAMPT P43490 1/20 0.35
GPR119 Q8TDV5 1/20 0.35
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
ENPP2 Q13822 1/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29563944 0.84 MBOAT4 (0.44) LMNAALDH1A1MBOAT4MAP4K4JAK2
SCHEMBL24612155 0.78 MBOAT4 (0.44) MBOAT4HTR2AHTR2CKCNH2LOX
SCHEMBL28536047 0.78 MBOAT4 (0.43) LMNAMBOAT4MAP4K4JAK2LOX
SCHEMBL3129623 0.77 LMNA (0.39) LMNAALDH1A1
SCHEMBL1851646 0.77 ADRA2A (0.41) ALDH1A1FFAR1
SCHEMBL568140 0.76 LOXL2 (0.47) MBOAT4HTR2AHTR2CKCNH2LOX
SCHEMBL23530021 0.76 PTGS2 (0.43) MBOAT4HTR2AHTR2CKCNH2MAP4K4
SCHEMBL18457325 0.76 PTGDR2 (0.45) LMNAMBOAT4NAMPTGPR119PTGS1
SCHEMBL2697225 0.75 KMT2A (0.47) ALDH1A1MAP4K4JAK2PTGS2ENPP2
SCHEMBL2653485 0.75 ALDH1A1 (0.64) LMNAALDH1A1PRMT1GSRENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2324028-A2 THERAPEUTIC AGENTS 414 AstraZeneca AB (SE) 2011-05-25 EP disclosed
WO-2010015849-A2 THERAPEUTIC AGENTS 414 ASTRAZENECA AB (SE) 2010-02-11 WO disclosed