SCHEMBL18533995

SCHEMBL18533995

C=Cc1cc(C)ccc1CNc1cc(Cl)nc(N2CCNCC2)n1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.39
CTSB P07858 1/20 0.39
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
ROCK2 O75116 3/20 0.38
PLK4 O00444 1/20 0.37
PAK4 O96013 1/20 0.37
CCR4 P51679 1/20 0.36
CTNNB1 P35222 2/20 0.36
TCF7L2 Q9NQB0 2/20 0.36
SRC P12931 1/20 0.35
PDE4A P27815 2/20 0.35
PDE4B Q07343 2/20 0.35
PDE4C Q08493 2/20 0.35
PDE4D Q08499 2/20 0.35
PKM P14618 1/20 0.35
SOS1 Q07889 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16258707 0.78 CCR4 (0.55) ACHECCR4
SCHEMBL18153389 0.73 ROCK2 (0.56) ROCK2SRC
SCHEMBL2366622 0.69 HTR1A (0.51)
SCHEMBL18063490 0.66 CASP1 (0.50) ROCK2PLK4PAK4PDE4APDE4B
SCHEMBL22616040 0.64 ALDH1A1 (0.53) ACHECTSBCTSSCTSKROCK2
SCHEMBL16258648 0.63 CCR4 (0.51) CCR4
SCHEMBL19295961 0.63 KDM4E (0.41) SRC
SCHEMBL9845815 0.63 KMT2A (0.40) SRC
SCHEMBL9085080 0.62 HRH4 (0.52) ACHEROCK2
SCHEMBL22542113 0.61 HTR3A (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2805947-B1 PIPERAZINYL PYRIMIDINE DERIVATIVES, PREPARATION METHOD AND USE THEREOF INST PHARMACOLOGY & TOXICOLOGY ACAD MILITARY MEDICAL SCIENCES PLA CHINA (CN) 2017-02-22 EP disclosed