SCHEMBL185449

SCHEMBL185449

O=C(O)Oc1cnc(O)nc1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.33
F2 P00734 1/20 0.33
GLA P06280 1/20 0.33
HPGD P15428 1/20 0.33
HCAR2 Q8TDS4 1/20 0.31
P4HTM Q9NXG6 1/20 0.31
GABRP O00591 1/20 0.30
GABRD O14764 1/20 0.30
GABRA1 P14867 1/20 0.30
GABRB1 P18505 1/20 0.30
GABRG2 P18507 1/20 0.30
GABRB3 P28472 1/20 0.30
GABRA5 P31644 1/20 0.30
GABRA3 P34903 1/20 0.30
GABRA2 P47869 1/20 0.30
GABRB2 P47870 1/20 0.30
GABRA4 P48169 1/20 0.30
GABRE P78334 1/20 0.30
GABRA6 Q16445 1/20 0.30
GABRG1 Q8N1C3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7020112 0.81 ALDH1A1 (0.33) ALDH1A1F2GLAHPGDHCAR2
SCHEMBL185620 0.79 LMNA (0.35) ALDH1A1F2GLAHPGDHCAR2
SCHEMBL186176 0.79 HDAC1 (0.42) ALDH1A1F2GLAHPGDHCAR2
SCHEMBL185725 0.79 NAAA (0.41)
SCHEMBL10646167 0.77 ALDH1A1 (0.38) ALDH1A1F2GLAHPGDP4HTM
SCHEMBL185995 0.76 ALDH1A1 (0.59) ALDH1A1F2GLAHPGDKDM4E
SCHEMBL185429 0.76 ALDH1A1 (0.40) ALDH1A1F2GLAHPGDKDM4E
SCHEMBL198068 0.74 CCNE1 (0.35) ALDH1A1F2GLAHPGDHCAR2
SCHEMBL186014 0.74 L3MBTL1 (0.34) ALDH1A1GLAHPGDKDM4EHSD17B10
SCHEMBL186008 0.74 GRM5 (0.39) ALDH1A1F2GLAHPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed
EP-2401256-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2012-01-04 EP disclosed
WO-2010097372-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed