SCHEMBL185773

SCHEMBL185773

NC(=O)c1cccc(CCl)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 7/20 0.57
MEP1B Q16820 1/20 0.51
F10 P00742 1/20 0.49
ADRA1D P25100 1/20 0.48
FOLH1 Q04609 1/20 0.48
OPRM1 P35372 1/20 0.47
OPRD1 P41143 1/20 0.47
OPRK1 P41145 1/20 0.47
KCNH2 Q12809 1/20 0.47
IDH1 O75874 1/20 0.47
TSHR P16473 2/20 0.46
POLB P06746 1/20 0.46
CYP3A4 P08684 1/20 0.46
MAPT P10636 1/20 0.46
CYP2C19 P33261 1/20 0.46
RECQL P46063 1/20 0.46
BLM P54132 1/20 0.46
PMP22 Q01453 1/20 0.46
HSD17B10 Q99714 1/20 0.46
TDP1 Q9NUW8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30955451 1.00 PARP1 (0.57) PARP1MEP1BF10ADRA1DFOLH1
Pyridine SCHEMBL2326387 0.88 PARP1 (0.46) PARP1MEP1BF10ADRA1DFOLH1
SCHEMBL5232156 0.85 PARP1 (0.53) PARP1MEP1BF10ADRA1DFOLH1
SCHEMBL17672270 0.83 PLA2G2A (0.59) PARP1MEP1BF10FOLH1IDH1
SCHEMBL46680 0.82 FOLH1 (0.66) MEP1BFOLH1MRGPRX4MEN1KMT2A
SCHEMBL509423 0.82 LOXL2 (0.66) PARP1MEP1BFOLH1IDH1TSHR
SCHEMBL29364575 0.82 LOXL2 (0.66) PARP1MEP1BFOLH1IDH1TSHR
SCHEMBL2734990 0.82 PRSS1 (0.66) PARP1MEP1BF10FOLH1IDH1
SCHEMBL39676 0.82 TSHR (0.47) FOLH1TSHRMRGPRX4
SCHEMBL28410476 0.82 FOLH1 (0.46) FOLH1TSHRL3MBTL1MRGPRX4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 172 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250388592-A1 (AZA)SPIROHEPTANE DERIVATIVES FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS REMYND N.V. (BE) 2025-12-25 US disclosed
WO-2025231152-A1 COMPOUNDS AND METHODS FOR RESTORING BETA-ADRENERGIC RECEPTOR FUNCTION THE CLEVELAND CLINIC FOUNDATION (US) 2025-11-06 WO disclosed
US-12428745-B2 Method and system for electroplating parts with metal DIPSOL CHEMICALS CO., LTD. (JP) 2025-09-30 US disclosed
EP-4568968-A1 (AZA)SPIROHEPTANE DERIVATIVES FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS Remynd N.V. (BE) 2025-06-18 EP disclosed
EP-4524295-A2 METHOD AND SYSTEM FOR ELECTROPLATING ARTICLE WITH METAL Dipsol Chemicals Co., Ltd. (JP) 2025-03-19 EP disclosed
US-20240392461-A1 METHOD AND SYSTEM FOR ELECTROPLATING ARTICLE WITH METAL DIPSOL CHEM (JP) 2024-11-28 US disclosed
WO-2024115667-A1 NON PEPTIDERGIC AGONISTS OF OXYTOCIN RECEPTOR UNIVERSITE DE STRASBOURG (FR) 2024-06-06 WO disclosed
WO-2024033479-A1 (AZA)SPIROHEPTANE DERIVATIVES FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS REMYND N.V. (BE) 2024-02-15 WO disclosed
US-20230349063-A1 Method and System for Electroplating Parts with Metal DIPSOL CHEMICALS CO., LTD. (JP) 2023-11-02 US disclosed
EP-4269663-A1 METHOD AND SYSTEM FOR ELECTROPLATING ARTICLE WITH METAL Dipsol Chemicals Co., Ltd. (JP) 2023-11-01 EP disclosed
US-20010007877-A1 NOVEL ANTI-INFECTIVES SMITHKLINE BEECHAM CORPORATION 2001-07-12 US disclosed
EP-1112251-A1 AZETIDINE DERIVATIVES, PREPARATION AND MEDICINES CONTAINING THEM Aventis Pharma S.A. (FR) 2001-07-04 EP disclosed
EP-1100797-A1 HETEROCYCLIC COMPOUNDS AS INHIBITORS OF ROTAMASE ENZYMES Pfizer Limited (GB) 2001-05-23 EP disclosed
WO-2001034146-A1 NOVEL ANTI-INFECTIVES SMITHKLINE BEECHAM CORPORATION (US) 2001-05-17 WO disclosed
EP-1047698-A1 PIPERAZINO DERIVATIVES AS NEUROKININ ANTAGONISTS SCHERING CORPORATION (US) 2000-11-02 EP disclosed
WO-2000032582-A1 BENZAMIDE DERIVATIVES AND THEIR USE AS APOB-100 SECRETION INHIBITORS GLAXO GROUP LIMITED (GB) 2000-06-08 WO disclosed
WO-2000015609-A1 AZETIDINE DERIVATIVES, PREPARATION AND MEDICINES CONTAINING THEM AVENTIS PHARMA S.A. (FR) 2000-03-23 WO disclosed
WO-2000005232-A1 HETEROCYCLIC COMPOUNDS AS INHIBITORS OF ROTAMASE ENZYMES PFIZER LIMITED (GB) 2000-02-03 WO disclosed
WO-1999036424-A1 PIPERAZINO DERIVATIVES AS NEUROKININ ANTAGONISTS SCHERING CORPORATION (US) 1999-07-22 WO disclosed
US-5332738-A Imidazolidine antipsychotic agents NCNEILAB, INC. (US) 1994-07-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010007877-A1 NOVEL ANTI-INFECTIVES CTSL, MMP8, SERPINB1 PARP1 3238/4885MEP1B 2340/4885F10 4127/4885
US-20250388592-A1 (AZA)SPIROHEPTANE DERIVATIVES FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS SNCA, CHRNA6, CHRNA5 PARP1 1195/4885MEP1B 1114/4885F10 4429/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.