SCHEMBL186339

SCHEMBL186339

N#Cc1ncc(F)cc1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN2 Q96KS0 2/20 0.42
CYP11B1 P15538 3/20 0.37
CYP11B2 P19099 3/20 0.37
ALDH1A1 P00352 3/20 0.34
KDM4E B2RXH2 1/20 0.34
POLB P06746 1/20 0.34
PIK3CD O00329 1/20 0.34
ABL1 P00519 1/20 0.34
GRM5 P41594 1/20 0.33
USP8 P40818 1/20 0.33
USP7 Q93009 1/20 0.33
USP47 Q96K76 1/20 0.33
ERBB2 P04626 1/20 0.32
TRPV4 Q9HBA0 1/20 0.32
JAK2 O60674 2/20 0.32
NTRK1 P04629 1/20 0.32
CDK2 P24941 1/20 0.32
STAT5B P51692 1/20 0.32
JAK3 P52333 1/20 0.32
AURKB Q96GD4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29929823 1.00 EGLN2 (0.42) EGLN2CYP11B1CYP11B2ALDH1A1KDM4E
SCHEMBL384105 0.78 KEAP1 (0.38) EGLN2CYP11B1CYP11B2ALDH1A1KDM4E
SCHEMBL16321670 0.78 ALDH1A1 (0.44) EGLN2CYP11B1CYP11B2ALDH1A1KDM4E
SCHEMBL1976471 0.78 ABL1 (0.35) EGLN2CYP11B1CYP11B2ALDH1A1KDM4E
SCHEMBL30834616 0.78 PIK3CD (0.51) EGLN2CYP11B1CYP11B2ALDH1A1KDM4E
SCHEMBL18109302 0.78 PIK3CD (0.51) EGLN2CYP11B1CYP11B2ALDH1A1KDM4E
SCHEMBL10325957 0.78 AGBL2 (0.41) EGLN2CYP11B1CYP11B2ALDH1A1KDM4E
SCHEMBL12721108 0.78 EGLN2 (0.40) EGLN2CYP11B1CYP11B2ALDH1A1KDM4E
SCHEMBL16769277 0.78 CYP11B1 (0.40) EGLN2CYP11B1CYP11B2ALDH1A1KDM4E
SCHEMBL2298550 0.78 EGLN2 (0.40) EGLN2CYP11B1CYP11B2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 420 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117199519-A Electrolyte, preparation method and application thereof, and lithium battery 北京纳米能源与系统研究所 2023-12-08 CN claimed
CN-114984928-A Modified porous cyclodextrin polymer material and preparation method and application thereof 中南大学 2022-09-02 CN claimed
CN-112300793-A Preparation method of pure organic phosphorescent material based on bis-carbazole pyridine derivative 北京化工大学 2021-02-02 CN claimed
EP-2069325-A2 ISOQUINOLINE, QUINAZOLINE AND PHTHALAZINE DERIVATIVES Serenex, Inc. (US) 2009-06-17 EP claimed
US-20080070935-A1 Isoquinoline, Quinazoline and Phthalazine Derivatives ESANEX, INC. 2008-03-20 US claimed
WO-2008024977-A2 ISOQUINOLINE, QUINAZOLINE AND PHTHALAZINE DERIVATIVES SERENEX, INC. (US) 2008-02-28 WO claimed
EP-4698520-A1 RAF-MEK PROTEIN COMPLEX MODULATORS AND METHODS OF USE THEREOF Gandeeva Therapeutics, Inc. (US) 2026-02-25 EP disclosed
EP-4688155-A1 MORPHOLINE OREXIN RECEPTOR ANTAGONISTS Bial-Portela & CA, S.A. (PT) 2026-02-11 EP disclosed
EP-4655284-A1 MICROBIOCIDAL PYRAZOLE DERIVATIVES Syngenta Crop Protection AG (CH) 2025-12-03 EP disclosed
WO-2025235874-A1 HETEROCYCLICS AS EGFR INHIBITORS SCHRÖDINGER, INC. (US) 2025-11-13 WO disclosed
WO-2025093624-A1 A PROCESS FOR PREPARING 3,5-DIFLUORO-2-PYRIDINECARBOXAMIDE INTERVET INTERNATIONAL B.V. (NL) 2025-05-08 WO disclosed
US-20250051347-A1 BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUND AND USE THEREOF AS ANDROGEN RECEPTOR DEGRADER Hinova Pharmaceuticals, Inc. (CN) 2025-02-13 US disclosed
WO-2025023852-A1 MORPHOLINE OREXIN RECEPTOR ANTAGONISTS BIAL - PORTELA & CA., S.A. (PT) 2025-01-30 WO disclosed
WO-2001068640-A1 MEDICAMENTS AGAINST VIRAL DISEASES BAYER AKTIENGESELLSCHAFT (DE) 2001-09-20 WO disclosed
WO-2001068641-A1 6-AMINOALKYL-DIHYDROPYRIMIDINES AND THE USE THEREOF AS MEDICAMENTS AGAINST VIRAL DISEASES BAYER AKTIENGESELLSCHAFT (DE) 2001-09-20 WO disclosed
WO-2001068642-A1 DIHYDROPYRIMIDINES AND THE USE THEREOF AS MEDICAMENTS FOR THE TREATMENT OF HEPATITIS B BAYER AKTIENGESELLSCHAFT (DE) 2001-09-20 WO disclosed
WO-2001068647-A1 MEDICAMENTS AGAINST VIRAL DISEASES BAYER AKTIENGESELLSCHAFT (DE) 2001-09-20 WO disclosed
EP-1080086-A1 DIHYDROPYRIMIDINES BAYER AG (DE) 2001-03-07 EP disclosed
WO-2000058302-A1 DIHYDROPYRIMIDINES AND THEIR USE IN THE TREATMENT OF HEPATITIS B BAYER AKTIENGESELLSCHAFT (DE) 2000-10-05 WO disclosed
WO-1999054326-A1 DIHYDROPYRIMIDINES BAYER AKTIENGESELLSCHAFT (DE) 1999-10-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080070935-A1 Isoquinoline, Quinazoline and Phthalazine Derivatives H1-5, NDUFS5, IL5 EGLN2 1843/4885CYP11B1 944/4885CYP11B2 921/4885
US-20250051347-A1 BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUND AND USE THEREOF AS ANDROGEN RECEPTOR DEGRADER AR, ADRM1, MDM2 EGLN2 4585/4885CYP11B1 194/4885CYP11B2 324/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.