SCHEMBL384105

SCHEMBL384105

N#Cc1ncc(F)cc1Br

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.38
HTT P42858 1/20 0.37
CYP11B1 P15538 3/20 0.37
CYP11B2 P19099 3/20 0.37
ABL1 P00519 1/20 0.33
PIK3CD O00329 1/20 0.33
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
GRM5 P41594 2/20 0.32
EGLN2 Q96KS0 2/20 0.31
USP8 P40818 1/20 0.31
USP7 Q93009 1/20 0.31
USP47 Q96K76 1/20 0.31
ERBB2 P04626 1/20 0.31
JAK2 O60674 1/20 0.30
NTRK1 P04629 1/20 0.30
CDK2 P24941 1/20 0.30
STAT5B P51692 1/20 0.30
JAK3 P52333 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4719121 0.78 KMT2A (0.46) HTTCYP11B1CYP11B2ABL1PIK3CD
SCHEMBL29929823 0.78 EGLN2 (0.42) CYP11B1CYP11B2ABL1PIK3CDKDM4E
SCHEMBL186339 0.78 EGLN2 (0.42) CYP11B1CYP11B2ABL1PIK3CDKDM4E
SCHEMBL22865157 0.77 HTT (0.38) HTTPIK3CDKDM4EALDH1A1POLB
SCHEMBL11031954 0.76 CYP11B1 (0.32) HTTCYP11B1CYP11B2
SCHEMBL1976471 0.75 ABL1 (0.35) CYP11B1CYP11B2ABL1PIK3CDKDM4E
SCHEMBL30834616 0.75 PIK3CD (0.51) HTTCYP11B1CYP11B2ABL1PIK3CD
SCHEMBL18109302 0.75 PIK3CD (0.51) HTTCYP11B1CYP11B2ABL1PIK3CD
SCHEMBL10325957 0.75 AGBL2 (0.41) CYP11B1CYP11B2ABL1PIK3CDKDM4E
SCHEMBL16321670 0.75 ALDH1A1 (0.44) HTTCYP11B1CYP11B2ABL1PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 90 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026098567-A1 MACROCYCLIC COMPOUNDS AND USE THEREOF 微境生物医药科技(上海)有限公司 2026-05-15 WO disclosed
US-20260115199-A1 TRICYCLIC COMPOUNDS FOR THE TREATMENT OF CANCER HOFFMANN-LA ROCHE INC. (US) 2026-04-30 US disclosed
US-12606541-B2 PPARg modulators and methods of use EISAI R&D MANAGEMENT CO., LTD. (JP) 2026-04-21 US disclosed
US-12600732-B2 Bifunctional compounds for degrading BTK via ubiquitin proteosome pathway NURIX THERAPEUTICS, INC. (US) 2026-04-14 US disclosed
US-12590089-B2 Processes for preparing toll-like receptor modulator compounds GILEAD SCIENCES, INC. (US) 2026-03-31 US disclosed
US-12565497-B2 Sulfone derivatives HOFFMANN-LA ROCHE INC. (US) 2026-03-03 US disclosed
US-12441754-B2 Galactoside inhibitor of galectins GALECTO BIOTECH AB (DK) 2025-10-14 US disclosed
EP-4570320-A2 BIFUNCTIONAL COMPOUNDS FOR DEGRADING BTK VIA UBIQUITIN PROTEOSOME PATHWAY Nurix Therapeutics, Inc. (US) 2025-06-18 EP disclosed
WO-2025087431-A1 PAN-KRAS INHIBITOR AND USE THEREOF IN MEDICINES 贝达药业股份有限公司 2025-05-01 WO disclosed
US-20250122195-A1 POLYHETEROCYCLIC COMPOUNDS AS METTL3 INHIBITORS STORM THERAPEUTICS LIMITED (GB) 2025-04-17 US disclosed
US-20140113931-A1 SUBSTITUTED PICOLINAMIDE KINASE INHIBITORS PORTOLA PHARMACEUTICALS, INC. (US) 2014-04-24 US disclosed
US-20140113931-A1 SUBSTITUTED PICOLINAMIDE KINASE INHIBITORS PORTOLA PHARMACEUTICALS, INC. (US) 2014-04-24 US disclosed
WO-2013052394-A1 2-PYRIDYL CARBOXAMIDE-CONTAINING SPLEEN TYROSINE KINASE (SYK) INHIBITORS MERCK SHARP & DOHME CORP. (US) 2013-04-11 WO disclosed
WO-2013052394-A1 2-PYRIDYL CARBOXAMIDE-CONTAINING SPLEEN TYROSINE KINASE (SYK) INHIBITORS MERCK SHARP & DOHME CORP. (US) 2013-04-11 WO disclosed
EP-2408762-A1 HSP90 INHIBITING INDAZOLE DERIVATIVES, COMPOSITIONS CONTAINING SAME AND USE THEREOF SANOFI (FR) 2012-01-25 EP disclosed
US-20120010241-A1 HSP90 INHIBITING INDAZOLE DERIVATIVES, COMPOSITIONS CONTAINING SAME AND USE THEREOF SANOFI (FR) 2012-01-12 US disclosed
WO-2011004132-A1 NOVEL HSP90-INHIBITING INDOLE DERIVATIVES, COMPOSITIONS CONTAINING SAID DERIVATIVES, AND USE THEREOF SANOFI-AVENTIS (FR) 2011-01-13 WO disclosed
WO-2010106290-A1 HSP90 INHIBITING INDAZOLE DERIVATIVES, COMPOSITIONS CONTAINING SAME AND USE THEREOF SANOFI-AVENTIS (FR) 2010-09-23 WO disclosed
CN-100494178-C Preparation method of pyridine formamidine and salt thereof DONGYANGGUANG PHARMACEUTICAL C (CN) 2009-06-03 CN disclosed
CN-101029023-A Preparation method of pyridine formamidine and salt thereof DONGYANGGUANG PHARMACEUTICAL C (CN) 2007-09-05 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120010241-A1 HSP90 INHIBITING INDAZOLE DERIVATIVES, COMPOSITIONS CONTAINING SAME AND USE THEREOF HSP90AB2P, HSP90AB1, HSP90AA1 KEAP1 1381/4885HTT 541/4885CYP11B1 345/4885
US-12590089-B2 Processes for preparing toll-like receptor modulator compounds TLR8, MYD88, TLR6 KEAP1 1034/4885HTT 4876/4885CYP11B1 2205/4885
US-20250122195-A1 POLYHETEROCYCLIC COMPOUNDS AS METTL3 INHIBITORS METTL3, DIMT1, TPMT KEAP1 1756/4885HTT 2970/4885CYP11B1 1405/4885
US-20260115199-A1 TRICYCLIC COMPOUNDS FOR THE TREATMENT OF CANCER H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, HCCS, CCR6 KEAP1 923/4885HTT 2868/4885CYP11B1 46/4885
US-20140113931-A1 SUBSTITUTED PICOLINAMIDE KINASE INHIBITORS SYK, LCK, BTK KEAP1 2373/4885HTT 3624/4885CYP11B1 4274/4885
US-12441754-B2 Galactoside inhibitor of galectins LGALS1, LGALS3, LGALS2 KEAP1 689/4885HTT 4827/4885CYP11B1 354/4885
US-12606541-B2 PPARg modulators and methods of use PPARG, PPARA, PPARD KEAP1 1980/4885HTT 1624/4885CYP11B1 18/4885
US-12600732-B2 Bifunctional compounds for degrading BTK via ubiquitin proteosome pathway BTK, BCL9, BCL9L KEAP1 1214/4885HTT 2260/4885CYP11B1 4111/4885
US-12565497-B2 Sulfone derivatives CXCR1, CCR1, SULT1E1 KEAP1 1045/4885HTT 3992/4885CYP11B1 44/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.