SCHEMBL18746522

SCHEMBL18746522

CCOC(=O)N1CCN(CCCc2ccc(-n3ccnc3)cc2)CC1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.71
CYP2C9 P11712 2/20 0.71
CYP1A2 P05177 1/20 0.71
CYP2C19 P33261 1/20 0.71
TBXAS1 P24557 2/20 0.53
HTR2A P28223 2/20 0.53
OPRM1 P35372 2/20 0.53
ADORA3 P0DMS8 1/20 0.53
HTR7 P34969 1/20 0.53
SIGMAR1 Q99720 1/20 0.53
HRH1 P35367 5/20 0.50
HRH2 P25021 4/20 0.50
LSS P48449 1/20 0.49
KDM4E B2RXH2 2/20 0.48
TSHR P16473 1/20 0.48
MAPK1 P28482 1/20 0.48
ATM Q13315 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
MEN1 O00255 1/20 0.48
MITF O75030 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14129949 0.83 CYP1A2 (1.00) CYP2D6CYP2C9CYP1A2CYP2C19HRH1
SCHEMBL11484688 0.78 TBXAS1 (0.68) CYP2D6CYP2C9CYP1A2CYP2C19TBXAS1
SCHEMBL9744374 0.77 ALDH1A1 (0.57) HTR2AOPRM1ADORA3HTR7SIGMAR1
SCHEMBL10508433 0.75 HRH2 (0.63) HTR2AOPRM1ADORA3HTR7SIGMAR1
SCHEMBL9819864 0.74 SIGMAR1 (0.69) CYP2C19HTR2AOPRM1ADORA3HTR7
Hydrochloric Acid SCHEMBL10509615 0.74 HRH1 (0.61) HTR2AOPRM1ADORA3HTR7SIGMAR1
SCHEMBL9523895 0.73 CYP2C19 (0.60) CYP2D6CYP2C9CYP1A2CYP2C19LSS
SCHEMBL7404987 0.73 MAPT (0.63) CYP2D6CYP2C9CYP1A2CYP2C19TBXAS1
SCHEMBL10562129 0.72 LSS (0.60) CYP2D6CYP2C9CYP1A2CYP2C19HRH1
SCHEMBL28108298 0.72 CYP3A4 (0.65) CYP2D6CYP2C9CYP1A2CYP2C19TBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2061450-B1 METHODS OF MODULATING CELL PROLIFERATION AND CYST FORMATION IN POLYCYSTIC KIDNEY AND LIVER DISEASES MEDICAL COLLEGE WISCONSIN INC (US) 2017-04-19 EP disclosed