SCHEMBL1907796

SCHEMBL1907796

CC/C(=C/c1ccc(F)c(Br)c1)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPEP1 P16444 2/20 0.49
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
MAOA P21397 4/20 0.42
MAOB P27338 4/20 0.42
TBXAS1 P24557 2/20 0.42
TRPA1 O75762 2/20 0.41
VCP P55072 1/20 0.41
PSEN1 P49768 1/20 0.40
PSEN2 P49810 1/20 0.40
APH1B Q8WW43 1/20 0.40
NCSTN Q92542 1/20 0.40
APH1A Q96BI3 1/20 0.40
PSENEN Q9NZ42 1/20 0.40
EPHX2 P34913 2/20 0.40
GABRA1 P14867 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
PPARG P37231 1/20 0.39
ESR1 P03372 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2394174 1.00 DPEP1 (0.49) DPEP1NPC1RAB9ATDP1MAOA
SCHEMBL9515290 0.86 TBXAS1 (0.48) DPEP1TBXAS1PSEN1PSEN2APH1B
SCHEMBL9515296 0.86 TBXAS1 (0.48) DPEP1TBXAS1PSEN1PSEN2APH1B
SCHEMBL16566603 0.83 TBXAS1 (0.43) DPEP1TBXAS1TRPA1PSEN1PSEN2
SCHEMBL2392661 0.83 KMT2A (0.47) TBXAS1ESR1
SCHEMBL2555924 0.82 TRPA1 (0.55) DPEP1NPC1RAB9ATBXAS1TRPA1
SCHEMBL2555923 0.82 TRPA1 (0.55) DPEP1NPC1RAB9ATBXAS1TRPA1
SCHEMBL2389154 0.79 PSEN1 (0.51) NPC1RAB9ATDP1PSEN1PSEN2
SCHEMBL5173409 0.78 TBXAS1 (0.58) TBXAS1EPHX2PPARGESR1GRIK1
SCHEMBL12499859 0.77 ALDH1A1 (0.41) NPC1TDP1TBXAS1PSEN1PSEN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2493845-B1 SUBSTITUTED 3-PHENYLPROPIONIC ACIDS AND THE USE THEREOF BAYER IP GMBH (DE) 2013-12-25 EP disclosed
EP-2493845-A1 SUBSTITUTED 3-PHENYLPROPIONIC ACIDS AND THE USE THEREOF Bayer Pharma Aktiengesellschaft (DE) 2012-09-05 EP disclosed
WO-2011051165-A1 SUBSTITUTED 3-PHENYLPROPIONIC ACIDS AND THE USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2011-05-05 WO disclosed