SCHEMBL19086212

SCHEMBL19086212

CC[C@@H](NC(=O)c1ccc2[nH]ncc2c1)C(=O)N1CCc2sc(CNCc3cccc(F)c3)cc2C1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 12/20 0.41
ROCK1 Q13464 9/20 0.41
MAPK1 P28482 1/20 0.38
NPC1 O15118 1/20 0.37
DYRK3 O43781 1/20 0.37
MAP4K4 O95819 1/20 0.37
RPS6KB1 P23443 1/20 0.37
CLK2 P49760 1/20 0.37
RAB9A P51151 1/20 0.37
CSNK2A1 P68400 1/20 0.37
DYRK1A Q13627 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
MKNK2 Q9HBH9 1/20 0.37
HCRTR2 O43614 3/20 0.36
HCRTR1 O43613 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19085994 0.89 ROCK2 (0.41) ROCK2ROCK1MAPK1SMN1; SMN2
SCHEMBL19085978 0.84 ROCK2 (0.46) ROCK2ROCK1NPC1DYRK3MAP4K4
SCHEMBL19085995 0.82 METTL3 (0.41) ROCK2ROCK1SMN1; SMN2KMT2A
SCHEMBL19085984 0.81 ROCK2 (0.42) ROCK2ROCK1HCRTR2SMN1; SMN2KMT2A
SCHEMBL19086023 0.81 NAMPT (0.38) ROCK2ROCK1
SCHEMBL19085976 0.81 DDR2 (0.46) ROCK2ROCK1
SCHEMBL19085996 0.80 ROCK2 (0.53) ROCK2ROCK1MAPK1DYRK3MAP4K4
SCHEMBL19085977 0.80 NPC1 (0.45) ROCK2ROCK1MAPK1NPC1DYRK3
SCHEMBL19086004 0.80 PRMT5 (0.39) ROCK2ROCK1NPC1RAB9A
SCHEMBL19086994 0.79 MAOB (0.39) ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed