SCHEMBL19088925

SCHEMBL19088925

COc1ccnc(C(=O)N[C@H]2COCC[C@@H](CC(C)(C)c3ccccc3)[C@H](C)OC2=O)c1O

nearest known ligand 0.31

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 3/20 0.31
TAS1R1 Q7RTX1 3/20 0.31
TAS1R2 Q8TE23 1/20 0.31
RIPK1 Q13546 1/20 0.30
ROCK2 O75116 1/20 0.30
ROCK1 Q13464 1/20 0.30
DRD2 P14416 1/20 0.30
GSK3A P49840 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19084208 0.90 TAS1R3 (0.36) TAS1R3TAS1R1TAS1R2DRD2
SCHEMBL19089228 0.88 ROCK1 (0.31) ROCK2ROCK1
SCHEMBL19088921 0.87 RIPK1 (0.36) TAS1R3TAS1R1TAS1R2RIPK1
SCHEMBL19088924 0.87 PDE4D (0.36) RIPK1
SCHEMBL19088927 0.86 TAS1R3 (0.33) TAS1R3TAS1R1TAS1R2RIPK1ROCK2
SCHEMBL19088918 0.85 PDE4D (0.34) TAS1R3TAS1R1TAS1R2
SCHEMBL17417044 0.84 RIPK1 (0.36) TAS1R3TAS1R1TAS1R2RIPK1
SCHEMBL19088919 0.84 PDE4D (0.34) TAS1R3TAS1R1TAS1R2
SCHEMBL17898894 0.82 HPGDS (0.32) TAS1R3TAS1R1TAS1R2RIPK1ROCK2
SCHEMBL19066904 0.82 GRM4 (0.34) RIPK1ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017116949-A1 MACROCYCLIC PICOLINAMIDES AS FUNGICIDES DOW AGROSCIENCES LLC (US) 2017-07-06 WO disclosed