SCHEMBL1921273

SCHEMBL1921273

CC(=O)On1ccc2ccc(N3CCNCC3)cc2c1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.42
HTR1D P28221 1/20 0.42
HTR1B P28222 1/20 0.42
HTR3E A5X5Y0 3/20 0.42
HTR3B O95264 3/20 0.42
HTR3A P46098 3/20 0.42
HTR3D Q70Z44 3/20 0.42
HTR3C Q8WXA8 3/20 0.42
SIGMAR1 Q99720 3/20 0.42
HTR5A P47898 2/20 0.42
ADRB1 P08588 9/20 0.40
ABHD6 Q9BV23 1/20 0.38
ABL1 P00519 1/20 0.37
PDK2 Q15119 1/20 0.37
HTR6 P50406 3/20 0.36
USP2 O75604 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
IDO1 P14902 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1920629 0.75 CYP3A4 (0.45) HTR1AHTR1DHTR1BHTR3EHTR3B
SCHEMBL3056753 0.73 HTR5A (0.43) HTR1AHTR1DHTR1BHTR3EHTR3B
SCHEMBL28499890 0.68 HTR3E (0.49) HTR1AHTR1DHTR1BHTR3EHTR3B
SCHEMBL4977907 0.67 HTR3E (0.59) HTR1AHTR1DHTR1BHTR3EHTR3B
SCHEMBL9396666 0.67 HTR3E (0.51) HTR1AHTR1DHTR1BHTR3EHTR3B
SCHEMBL7369557 0.65 HTR3E (0.49) HTR1AHTR1DHTR1BHTR3EHTR3B
SCHEMBL4543250 0.65 ADRB1 (0.62) HTR1AHTR1DHTR1BHTR3EHTR3B
SCHEMBL6964245 0.65 ADRB1 (0.65) HTR1AHTR3EHTR3BHTR3AHTR3D
SCHEMBL8705185 0.64 HTR1A (0.49) HTR1AHTR1DHTR1BHTR3EHTR3B
SCHEMBL12004436 0.64 HTR3E (0.54) HTR1AHTR1DHTR1BHTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2326666-A1 NEUROPEPTIDE-2 RECEPTOR (Y-2R) AGONISTS AND USES THEREOF F. Hoffmann-La Roche AG (CH) 2011-06-01 EP claimed
WO-2010031707-A1 NEUROPEPTIDE-2 RECEPTOR (Y-2R) AGONISTS AND USES THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2010-03-25 WO claimed