SCHEMBL19520187

SCHEMBL19520187

O=C(Nc1cncnc1)c1cccnc1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.81
HIF1A Q16665 1/20 0.81
ROCK2 O75116 1/20 0.73
ROCK1 Q13464 1/20 0.73
BCAT2 O15382 1/20 0.72
NAMPT P43490 3/20 0.68
TDP1 Q9NUW8 1/20 0.65
KCNK3 O14649 1/20 0.65
PIM1 P11309 1/20 0.63
PIM3 Q86V86 1/20 0.63
PIM2 Q9P1W9 1/20 0.63
RAB9A P51151 5/20 0.61
NPC1 O15118 4/20 0.61
SMN1; SMN2 Q16637 3/20 0.61
KMT2A Q03164 2/20 0.61
MEN1 O00255 1/20 0.61
ALDH1A1 P00352 1/20 0.61
TP53 P04637 1/20 0.61
HDAC1 Q13547 1/20 0.61
HDAC6 Q9UBN7 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1571386 0.89 LMNA (1.00) LMNAHIF1AROCK2ROCK1NAMPT
Nicotinanilide SCHEMBL352439 0.84 LMNA (0.83) LMNAHIF1AROCK2ROCK1NAMPT
SCHEMBL14880208 0.84 ROCK2 (1.00) LMNAHIF1AROCK2ROCK1NAMPT
Nicotinanilide SCHEMBL29067673 0.84 LMNA (0.83) LMNAHIF1AROCK2ROCK1NAMPT
SCHEMBL4243217 0.84 BCAT2 (1.00) LMNAHIF1ABCAT2NAMPTKCNK3
SCHEMBL1971026 0.83 NAMPT (0.78) LMNAHIF1AROCK2ROCK1NAMPT
Nicotinanilide SCHEMBL8155304 0.83 LMNA (0.81) LMNAHIF1AROCK2ROCK1NAMPT
SCHEMBL5384036 0.81 ROCK2 (0.76) LMNAHIF1AROCK2ROCK1NAMPT
SCHEMBL26429188 0.81 LMNA (0.71) LMNAHIF1AROCK2ROCK1NAMPT
SCHEMBL167081 0.81 NAMPT (1.00) LMNAHIF1ABCAT2NAMPTKCNK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017186148-A1 NOVEL HETEROCYCLIC COMPOUNDS AS TYROSINE KINASE BCR-ABL INHIBITORS ASTAR BIOTECH LLC (US) 2017-11-02 WO disclosed