SCHEMBL19558149

SCHEMBL19558149

Fc1ccc(-c2nnc(S)o2)cc1

nearest known ligand 0.72

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.72
RAB9A P51151 5/20 0.72
TSHR P16473 2/20 0.60
TP53 P04637 2/20 0.60
SMN1; SMN2 Q16637 2/20 0.60
HSD17B10 Q99714 1/20 0.60
USP2 O75604 1/20 0.58
POLB P06746 1/20 0.58
MAOA P21397 2/20 0.51
MAOB P27338 2/20 0.51
ACHE P22303 1/20 0.47
KDM4E B2RXH2 1/20 0.47
NOTUM Q6P988 2/20 0.47
ADCY1 Q08828 2/20 0.46
CHRNA7 P36544 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2289115 0.84 NPC1 (1.00) NPC1RAB9ATSHRTP53SMN1; SMN2
SCHEMBL9058872 0.79 NPC1 (0.60) NPC1RAB9ATSHRTP53SMN1; SMN2
SCHEMBL28628120 0.79 DGAT1 (0.60) NPC1RAB9ATSHRTP53SMN1; SMN2
SCHEMBL7724942 0.79 RAB9A (0.72) NPC1RAB9ATP53SMN1; SMN2HSD17B10
SCHEMBL9364714 0.79 ACHE (0.47) NPC1RAB9ATP53SMN1; SMN2USP2
SCHEMBL988353 0.79 NPC1 (0.62) NPC1RAB9ATSHRTP53SMN1; SMN2
SCHEMBL28353634 0.79 NPC1 (0.64) NPC1RAB9ATP53SMN1; SMN2HSD17B10
SCHEMBL21434668 0.79 NOTUM (0.47) NPC1RAB9ATSHRTP53SMN1; SMN2
SCHEMBL6296345 0.79 NPC1 (0.55) NPC1RAB9ATP53SMN1; SMN2HSD17B10
SCHEMBL406885 0.78 NPC1 (0.70) NPC1RAB9ATSHRTP53SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113461630-B Nootkatone thioether derivative containing 1,3, 4-oxadiazole ring, and preparation method and application thereof 郑州大学 2022-09-02 CN claimed
CN-113461630-A Nootkatone thioether derivative containing 1,3, 4-oxadiazole ring, and preparation method and application thereof 郑州大学 2021-10-01 CN claimed
CN-113582983-B 1,3,4-oxadiazole thioether myricetin derivative, preparation method and application 贵州大学 2023-04-18 CN disclosed
CN-113461630-B Nootkatone thioether derivative containing 1,3, 4-oxadiazole ring, and preparation method and application thereof 郑州大学 2022-09-02 CN disclosed
CN-113582983-A Myricetin derivative of 1,3, 4-oxadiazole thioether, preparation method and application 贵州大学 2021-11-02 CN disclosed
CN-113461630-A Nootkatone thioether derivative containing 1,3, 4-oxadiazole ring, and preparation method and application thereof 郑州大学 2021-10-01 CN disclosed
CN-105949181-B 4- hydroxypyrrole quinoline -2- ketone derivatives, preparation method and the application of the oxadiazoles containing 1,3,4- 贵州大学 2019-08-02 CN disclosed
US-9809545-B2 Factor XIa inhibitors MERCK SHARP & DOHME CORP. (US) 2017-11-07 US disclosed
CN-104292224-A Benzothiazole amide derivatives containing substituted 1,3,4-thiadiazole (oxadiazole) thioether as well as preparation method and application of derivatives UNIV GUIZHOU 2015-01-21 CN disclosed