SCHEMBL19622290

SCHEMBL19622290

CCCC(=O)c1ccc(Oc2ccc(P)c(CO)c2)nc1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 2/20 0.41
OPRM1 P35372 7/20 0.38
OPRD1 P41143 6/20 0.38
HRH3 Q9Y5N1 6/20 0.38
OPRK1 P41145 5/20 0.38
STS P08842 1/20 0.37
PDE4A P27815 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
MAPT P10636 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19622278 0.93 OPRM1 (0.41) PDE4BOPRM1OPRD1HRH3OPRK1
SCHEMBL19622279 0.74 HRH3 (0.38) PDE4BOPRM1OPRD1HRH3OPRK1
SCHEMBL19622337 0.71 LMNA (0.50) PDE4BOPRM1OPRD1OPRK1MAPT
SCHEMBL19622338 0.70 LMNA (0.49) PDE4BOPRM1OPRD1OPRK1MAPT
SCHEMBL19622328 0.69 PDE4B (0.44) PDE4BOPRM1OPRD1STSPDE4D
SCHEMBL19622283 0.68 MAPT (0.45) OPRM1OPRD1HRH3OPRK1MAPT
SCHEMBL19622334 0.68 P2RX3 (0.41)
SCHEMBL24376943 0.67 KDM4E (0.56) OPRM1OPRD1HRH3OPRK1MAPT
SCHEMBL9607407 0.66 HRH3 (0.58) HRH3L3MBTL1
SCHEMBL19622288 0.66 CYP4F2 (0.41) PDE4BOPRM1OPRD1HRH3OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3246034-A1 BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS Anacor Pharmaceuticals, Inc. (US) 2017-11-22 EP disclosed