SCHEMBL19634728

SCHEMBL19634728

CC(=O)NCc1cccc(C(=O)NCC(=O)NC(C)=C=O)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 2/20 0.45
HDAC2 Q92769 2/20 0.44
HDAC8 Q9BY41 2/20 0.44
HDAC6 Q9UBN7 2/20 0.44
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC9 Q9UKV0 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44
PPARG P37231 1/20 0.43
NR1H4 Q96RI1 1/20 0.43
ROCK2 O75116 4/20 0.41
LMNA P02545 1/20 0.41
HPGD P15428 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19634824 0.83 HTT (0.52) MMP13HDAC2HDAC8HDAC6HDAC3
SCHEMBL19634818 0.79 KDM1A (0.52) MMP13HDAC2HDAC8HDAC6HDAC3
SCHEMBL19634746 0.77 MMP13 (0.49) MMP13HDAC2HDAC8HDAC6HDAC3
SCHEMBL19634740 0.76 LOXL2 (0.64) MMP13HDAC2HDAC8HDAC6HDAC3
SCHEMBL19634801 0.76 SLC7A5 (0.58) MMP13HDAC2HDAC8HDAC6HDAC3
SCHEMBL16380331 0.75 ROCK2 (0.53) MMP13HDAC2HDAC8HDAC6HDAC3
SCHEMBL8646446 0.74 HDAC1 (0.57) MMP13HDAC2HDAC8HDAC6HDAC3
SCHEMBL19634816 0.73 ROCK2 (0.57) MMP13HDAC2HDAC8HDAC6HDAC3
SCHEMBL3530258 0.72 KMT2A (0.64) MMP13HDAC2HDAC8HDAC6HDAC3
SCHEMBL19634802 0.72 PARP1 (0.53) MMP13HDAC2HDAC8HDAC6HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017200984-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T GLOBAL INC. (US) 2017-11-23 WO disclosed