SCHEMBL19647775

SCHEMBL19647775

CCCCc1ccc(OC2C=CC(N)=CN2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 1/20 0.41
CRBN Q96SW2 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.38
CA2 P00918 3/20 0.38
NAAA Q02083 3/20 0.35
NPC1 O15118 1/20 0.35
TP53 P04637 1/20 0.35
TSHR P16473 1/20 0.35
RAB9A P51151 1/20 0.35
SKP2 Q13309 1/20 0.35
HTR2A P28223 1/20 0.34
CA1 P00915 1/20 0.33
THRB P10828 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
ALOX12 P18054 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2089333 0.66 DDB1 (0.45) DDB1CRBNSMN1; SMN2CA2NAAA
SCHEMBL27914349 0.65 CALM1 (0.68) SMN1; SMN2MEN1ALDH1A1LMNAGAA
SCHEMBL145761 0.65 LTA4H (0.52) SMN1; SMN2CA2TP53HTR2ACA1
SCHEMBL6558445 0.65 ALDH1A1 (0.54) SMN1; SMN2CA2NPC1TSHRRAB9A
SCHEMBL83869 0.64 CA2 (0.65) SMN1; SMN2CA2TP53SKP2HTR2A
SCHEMBL16933991 0.63 LMNA (0.62) SMN1; SMN2TSHRMEN1ALDH1A1LMNA
SCHEMBL145506 0.63 CALM1 (0.64) SMN1; SMN2MEN1ALDH1A1LMNAGAA
SCHEMBL111607 0.62 GFER (0.62) SMN1; SMN2CA2NPC1TP53TSHR
SCHEMBL13348593 0.62 POLB (0.50) SMN1; SMN2CA2NPC1TP53RAB9A
SCHEMBL5614714 0.62 LTA4H (0.66) TSHRALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2793884-B1 INHIBITORS OF NOTCH SIGNALLING PATHWAY AND USE THEREOF IN TREATMENT OF CANCERS ECOLE POLYTECHNIQUE FED LAUSANNE EPFL (CH) 2017-11-29 EP disclosed