SCHEMBL19657376

SCHEMBL19657376

C=CN(C)c1cc(Br)ccc1N(C)C

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 1/20 0.36
PYCR1 P32322 1/20 0.33
APP P05067 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
POLB P06746 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10187266 0.81 HRH4 (0.36) PYCR1ALDH1A1LMNAMAPK1
SCHEMBL7526844 0.74 ERN1 (0.34) CCR5PYCR1APPALDH1A1LMNA
SCHEMBL22272311 0.70 CCR5 (0.48) CCR5PYCR1APPALDH1A1HTT
SCHEMBL9485990 0.70 CCR5 (0.42) CCR5PYCR1APPALDH1A1POLB
SCHEMBL9566865 0.70 ALOX15 (0.42) CCR5PYCR1APPALDH1A1LMNA
SCHEMBL19657347 0.69 NMT1 (0.32)
SCHEMBL18228396 0.69 CCR5 (0.41) CCR5PYCR1APPALDH1A1LMNA
SCHEMBL14808309 0.69 HRH4 (0.41) CCR5PYCR1APPALDH1A1GAA
SCHEMBL24094415 0.68 HRH4 (0.33) CCR5PYCR1
SCHEMBL22339987 0.68 PYCR1 (0.33) PYCR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017205536-A2 THERAPEUTIC COMPOUNDS AND USES THEREOF GENENTECH, INC. (US) 2017-11-30 WO disclosed