SCHEMBL7526844

SCHEMBL7526844

C=Cc1cc(Br)ccc1N(C)C

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.34
PYCR1 P32322 1/20 0.34
CCR5 P51681 1/20 0.34
APP P05067 3/20 0.33
CA12 O43570 1/20 0.33
CA9 Q16790 1/20 0.33
ALDH1A1 P00352 4/20 0.32
GAA P10253 2/20 0.32
MAPT P10636 2/20 0.32
LMNA P02545 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
HPGD P15428 2/20 0.32
POLB P06746 1/20 0.32
MAPK1 P28482 1/20 0.32
TSHR P16473 1/20 0.30
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22339987 0.85 PYCR1 (0.33) ERN1PYCR1CA12CA9ALDH1A1
SCHEMBL23175927 0.82 ALDH1A3 (0.36) ERN1PYCR1CCR5ALDH1A1GAA
SCHEMBL2048237 0.80 CYP2A6 (0.38) PYCR1CCR5APPALDH1A1MAPT
SCHEMBL3209434 0.80 ERN1 (0.52) ERN1CCR5APPALDH1A1GAA
SCHEMBL31457111 0.80 ERN1 (0.52) ERN1CCR5APPALDH1A1GAA
SCHEMBL24633833 0.78 TP53 (0.38) APPALDH1A1GAAMAPTLMNA
SCHEMBL19657376 0.74 CCR5 (0.36) PYCR1CCR5APPALDH1A1GAA
SCHEMBL16953358 0.72 ERN1 (0.38) ERN1CA12CA9ALDH1A1GAA
SCHEMBL9566865 0.72 ALOX15 (0.42) PYCR1CCR5APPALDH1A1GAA
SCHEMBL2787330 0.72 HSP90AA1 (0.41) ERN1CA12CA9ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021057190-A1 QUINOLINE COMPOUNDS, PREPARATION METHOD THEREFOR AND USE THEREOF 上海阳帆医药科技有限公司 2021-04-01 WO disclosed
EP-0907684-B1 CROSS-LINKED SILICONE BASED MATERIAL COMPRISING A BOUND PHOTOINITIATOR, ITS METHOD OF PREPARATION, HYDROPHILIC POLYMERIC PRODUCT OBTAINED FROM THIS MATERIAL AND ITS METHOD OF PREPARATION, AND NOVEL PHOTOINITIATORS ESSILOR INT (FR) 2002-03-27 EP disclosed
US-20010007880-A1 Material based on crosslinked silicone polymer comprising an immobilized photoinitiator, process for the preparation thereof, hydrophilic polymeric product obtained from this material and process for the preparation thereof, and novel photoinitiators ESSILOR INTERNATIONAL COMPAGNIE GENERALE D'OPTIQUE 2001-07-12 US disclosed
US-6197842-B1 CONTACT LENSES ESSILOR INTERNATIONAL COMPAGNIE GENERALE D'OPTIQUE (FR) 2001-03-06 US disclosed
EP-0907684-A1 CROSS-LINKED SILICONE BASED MATERIAL COMPRISING A BOUND PHOTOINITIATOR, ITS METHOD OF PREPARATION, HYDROPHILIC POLYMERIC PRODUCT OBTAINED FROM THIS MATERIAL AND ITS METHOD OF PREPARATION, AND NOVEL PHOTOINITIATORS ESSILOR INTERNATIONAL COMPAGNIE GENERALE D'OPTIQUE (FR) 1999-04-14 EP disclosed
WO-1997049768-A1 CROSS-LINKED SILICONE BASED MATERIAL COMPRISING A BOUND PHOTOINITIATOR, ITS METHOD OF PREPARATION, HYDROPHILIC POLYMERIC PRODUCT OBTAINED FROM THIS MATERIAL AND ITS METHOD OF PREPARATION, AND NOVEL PHOTOINITIATORS ESSILOR INTERNATIONAL - COMPAGNIE GENERALE D'OPTIQUE (FR) 1997-12-31 WO disclosed