SCHEMBL19682803

SCHEMBL19682803

Cc1c(Cl)ccc(F)c1C=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
TDP1 Q9NUW8 2/20 0.41
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
HSD17B10 Q99714 1/20 0.33
MAPT P10636 1/20 0.33
RECQL P46063 1/20 0.32
PTGS2 P35354 3/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
LMNA P02545 2/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CES1 P23141 1/20 0.32
ERN1 O75460 1/20 0.31
VDR P11473 1/20 0.31
PTGS1 P23219 1/20 0.31
NPC1 O15118 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19682346 0.82 CYP2C9 (0.40) ALDH1A1MEN1KMT2ATDP1CYP3A4
SCHEMBL29954742 0.82 CYP2C9 (0.40) ALDH1A1MEN1KMT2ATDP1CYP3A4
SCHEMBL6663239 0.82 ALDH1A1 (0.54) ALDH1A1MEN1KMT2ATDP1HSD17B10
SCHEMBL12384956 0.78 ERN1 (0.38) ALDH1A1MEN1KMT2ATDP1CYP3A4
SCHEMBL29628640 0.78 ERN1 (0.38) ALDH1A1MEN1KMT2ATDP1CYP3A4
SCHEMBL615646 0.78 ALDH1A1 (0.44) ALDH1A1MEN1KMT2ATDP1CYP3A4
SCHEMBL953875 0.78 ALDH1A1 (0.44) ALDH1A1MEN1KMT2ATDP1CYP3A4
SCHEMBL29447959 0.78 ALDH1A1 (0.44) ALDH1A1MEN1KMT2ATDP1CYP3A4
SCHEMBL10290089 0.75 CYP3A4 (0.36) ALDH1A1MEN1KMT2ACYP3A4CYP2C9
SCHEMBL15748351 0.75 ERN1 (0.38) ALDH1A1CYP3A4CYP2C9CYP2C19ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10889555-B2 Sulfonamide compound or salt thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2021-01-12 US disclosed
US-20200405697-A1 Antitumor Agent TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-12-31 US disclosed
US-20200399235-A1 Sulfonamide Compound or Salt Thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-12-24 US disclosed
US-20200361883-A1 Sulfonamide Compounds and Use Thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-11-19 US disclosed
EP-3718545-A1 ANTITUMOR AGENT Taiho Pharmaceutical Co., Ltd. (JP) 2020-10-07 EP disclosed
US-20200157066-A1 Sulfonamide Compound or Salt Thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-05-21 US disclosed
EP-3466934-A1 SULFONAMIDE COMPOUND OR SALT THEREOF Taiho Pharmaceutical Co., Ltd. (JP) 2019-04-10 EP disclosed
WO-2017209155-A1 SULFONAMIDE COMPOUND OR SALT THEREOF 大鵬薬品工業株式会社 2017-12-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200399235-A1 Sulfonamide Compound or Salt Thereof RNASEH1, SNRPA1, RRM2 ALDH1A1 1103/4885MEN1 4320/4885KMT2A 869/4885
US-20200157066-A1 Sulfonamide Compound or Salt Thereof RNASEH1, SNRPA1, RRM2 ALDH1A1 1103/4885MEN1 4320/4885KMT2A 869/4885
US-20200361883-A1 Sulfonamide Compounds and Use Thereof STS, SULT2A1, TPST2 ALDH1A1 2960/4885MEN1 3504/4885KMT2A 2512/4885
US-10889555-B2 Sulfonamide compound or salt thereof RNASEH1, SNRPA1, RRM2 ALDH1A1 1103/4885MEN1 4320/4885KMT2A 869/4885
US-20200405697-A1 Antitumor Agent HNRNPR, RRM2, RRM2B ALDH1A1 1397/4885MEN1 3770/4885KMT2A 1647/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.