SCHEMBL1978497

SCHEMBL1978497

CCCNn1c(C)c(C(=O)NCC2(c3cccc(Cl)c3)CC2)c(C)c(Br)c1=O

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNA3 P22001 1/20 0.43
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
P2RX7 Q99572 5/20 0.37
SLC6A9 P48067 5/20 0.36
KCNH2 Q12809 2/20 0.36
IDO1 P14902 1/20 0.36
CACNA1I Q9P0X4 1/20 0.35
MCHR1 Q99705 2/20 0.34
TP53 P04637 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CNR1 P21554 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1979905 0.89 P2RX7 (0.43) KCNA3SLC6A2SLC6A4SLC6A3P2RX7
SCHEMBL10150960 0.82 PDE10A (0.42) SMN1; SMN2P2RX7TP53MEN1KMT2A
SCHEMBL2015522 0.79 BCL2 (0.42) ALDH1A1SMN1; SMN2TP53MEN1KMT2A
SCHEMBL10150652 0.75 THRB (0.50) ALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL1973915 0.75 PPARG (0.37)
SCHEMBL2013388 0.73 THRB (0.39) ALDH1A1
SCHEMBL10150590 0.72 PDE10A (0.42) GAAKMT2A
SCHEMBL2010877 0.71 L3MBTL1 (0.48) ALDH1A1GAASMN1; SMN2MEN1KMT2A
SCHEMBL1975060 0.69 PPARG (0.40) ALDH1A1SMN1; SMN2NPSR1TP53MEN1
SCHEMBL1973564 0.67 TACR3 (0.46) ALDH1A1SMN1; SMN2NPSR1TP53MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110144164-A1 Pyridone derivatives as NK3 antagonists H. LUNDBECK A/S (DK) 2011-06-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110144164-A1 Pyridone derivatives as NK3 antagonists KCNK3, GRIK3, KCND3 KCNA3 4/4885SLC6A2 218/4885SLC6A4 223/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.