SCHEMBL19869980

SCHEMBL19869980

COc1cc(B2OC(C)(C)C(C)(C)O2)cc(OC)c1CN(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD9 Q9H8M2 8/20 0.38
BRD4 O60885 6/20 0.38
BRD7 Q9NPI1 6/20 0.38
BRD2 P25440 4/20 0.38
CSF1R P07333 1/20 0.36
LPL P06858 6/20 0.35
LIPG Q9Y5X9 6/20 0.35
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 1/20 0.34
ACHE P22303 1/20 0.34
TAF1 P21675 1/20 0.33
TGFBR1 P36897 1/20 0.33
BRPF1 P55201 1/20 0.33
ACVR1 Q04771 1/20 0.33
BPTF Q12830 1/20 0.33
TAF1L Q8IZX4 1/20 0.33
CREBBP Q92793 1/20 0.33
CECR2 Q9BXF3 1/20 0.33
BAZ2B Q9UIF8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23629064 0.83 LIPG (0.34) CSF1RLPLLIPGMEN1ALDH1A1
SCHEMBL19747751 0.81 CD274 (0.43) CSF1RLPLLIPG
SCHEMBL27159855 0.79 ALDH1A1 (0.44) CSF1RLPLLIPGMEN1ALDH1A1
SCHEMBL24556542 0.79 BRD9 (0.37) BRD9BRD4BRD7BRD2MEN1
SCHEMBL23575590 0.78 USP30 (0.38) CSF1R
SCHEMBL23590154 0.76 AAK1 (0.33)
SCHEMBL19747728 0.76 AAK1 (0.37) CSF1R
SCHEMBL22726982 0.76 CSF1R (0.43) CSF1RLPLLIPGMEN1KMT2A
SCHEMBL2278746 0.76 ACHE (0.43) CSF1RLPLLIPGMEN1ALDH1A1
SCHEMBL20600668 0.75 CA1 (0.40) CSF1RLPLLIPGKMT2ASNCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12528825-B2 Compounds and uses thereof FOGHORN THERAPEUTICS INC. (US) 2026-01-20 US disclosed
US-12384776-B2 Compounds and uses thereof FOGHORN THERAPEUTICS INC. (US) 2025-08-12 US disclosed
US-20240150328-A1 METHODS AND COMPOUNDS FOR TREATING DISORDERS FOGHORN THERAPEUTICS INC. 2024-05-09 US disclosed
US-11773085-B2 Methods and compounds for treating disorders FOGHORN THERAPEUTICS INC. (US) 2023-10-03 US disclosed
US-11773085-B2 Methods and compounds for treating disorders FOGHORN THERAPEUTICS INC. (US) 2023-10-03 US disclosed
US-11773085-B2 Methods and compounds for treating disorders FOGHORN THERAPEUTICS INC. (US) 2023-10-03 US disclosed
US-20230072053-A1 COMPOUNDS AND USES THEREOF FOGHORN THERAPEUTICS INC. 2023-03-09 US disclosed
EP-3265453-B1 NEW PYRIDINONES AND ISOQUINOLINONES AS INHIBITORS OF THE BROMODOMAIN BRD9 BOEHRINGER INGELHEIM INT (DE) 2022-06-29 EP disclosed
EP-3265453-B1 NEW PYRIDINONES AND ISOQUINOLINONES AS INHIBITORS OF THE BROMODOMAIN BRD9 BOEHRINGER INGELHEIM INT (DE) 2022-06-29 EP disclosed
US-11319318-B2 Pyridinones and isoquinolinones as inhibitors of the bromodomain BRD9 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2022-05-03 US disclosed
EP-3917529-A1 COMPOUNDS AND USES THEREOF Foghorn Therapeutics Inc. (US) 2021-12-08 EP disclosed
WO-2021155100-A1 COMPOUNDS AND USES THEREOF FOGHORN THERAPEUTICS INC. (US) 2021-08-05 WO disclosed
US-20210009568-A1 METHODS AND COMPOUNDS FOR TREATING DISORDERS FOGHORN THERAPEUTICS INC. 2021-01-14 US disclosed
US-20210009568-A1 METHODS AND COMPOUNDS FOR TREATING DISORDERS FOGHORN THERAPEUTICS INC. 2021-01-14 US disclosed
EP-3746135-A1 METHODS AND COMPOUNDS FOR TREATING DISORDERS Foghorn Therapeutics Inc. (US) 2020-12-09 EP disclosed
WO-2020160196-A1 COMPOUNDS AND USES THEREOF FOGHORN THERAPEUTICS INC. (US) 2020-08-06 WO disclosed
WO-2019152440-A1 METHODS AND COMPOUNDS FOR TREATING DISORDERS FOGHORN THERAPEUTICS INC. (US) 2019-08-08 WO disclosed
WO-2019152440-A1 METHODS AND COMPOUNDS FOR TREATING DISORDERS FOGHORN THERAPEUTICS INC. (US) 2019-08-08 WO disclosed
US-20180044335-A1 New Pyridinones and Isoquinolinones as Inhibitors of the Bromodomain BRD9 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2018-02-15 US disclosed
US-20180044335-A1 New Pyridinones and Isoquinolinones as Inhibitors of the Bromodomain BRD9 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2018-02-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12384776-B2 Compounds and uses thereof VHL, TFEB, BECN1 BRD9 290/4885BRD4 42/4885BRD7 149/4885
US-20180044335-A1 New Pyridinones and Isoquinolinones as Inhibitors of the Bromodomain BRD9 BRD9, BRD1, BRD2 BRD9 1/4885BRD4 5/4885BRD7 6/4885
US-11319318-B2 Pyridinones and isoquinolinones as inhibitors of the bromodomain BRD9 BRD9, BRD1, BRD2 BRD9 1/4885BRD4 6/4885BRD7 5/4885
US-11773085-B2 Methods and compounds for treating disorders VHL, TFEB, BECN1 BRD9 330/4885BRD4 57/4885BRD7 263/4885
US-20240150328-A1 METHODS AND COMPOUNDS FOR TREATING DISORDERS VHL, TFEB, BECN1 BRD9 330/4885BRD4 57/4885BRD7 263/4885
US-12528825-B2 Compounds and uses thereof BRD9, BRD8, BRIX1 BRD9 1/4885BRD4 20/4885BRD7 21/4885
US-20230072053-A1 COMPOUNDS AND USES THEREOF VHL, CLN6, TFEB BRD9 434/4885BRD4 111/4885BRD7 156/4885
US-20210009568-A1 METHODS AND COMPOUNDS FOR TREATING DISORDERS VHL, TFEB, BECN1 BRD9 330/4885BRD4 57/4885BRD7 263/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.