Water

Water

SCHEMBL1989477

O.O=C(O)C(c1ccccc1Cl)N1CCc2sccc2C1

nearest known ligand 0.76

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Water. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 known ✓ P35372 3/20 0.76
ADRA2A known ✓ P08913 2/20 0.76
OPRK1 known ✓ P41145 2/20 0.76
HTR2B known ✓ P41595 2/20 0.76
CHRM2 known ✓ P08172 2/20 0.76
THRB known ✓ P10828 1/20 0.76
HTR2A known ✓ P28223 1/20 0.76
SLC6A4 known ✓ P31645 1/20 0.76
ADORA3 known ✓ P0DMS8 2/20 0.46
ADRB3 known ✓ P13945 1/20 0.46
ADRA2B known ✓ P18089 1/20 0.46
ADRA2C known ✓ P18825 1/20 0.46
DRD4 known ✓ P21917 1/20 0.46
ADRA1A known ✓ P35348 1/20 0.46
DRD3 known ✓ P35462 1/20 0.46
SIGMAR1 known ✓ Q99720 1/20 0.46
ITGB3 known ✓ P05106 1/20 0.41
ITGA2B known ✓ P08514 1/20 0.41
CACNA2D1 known ✓ P54289 3/20 0.40
CACNA1B known ✓ Q00975 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL3377943 1.00 ABCB11 (0.76) ABCB11OPRM1CYP2C19ADRA2ACYP2B6
Hydrochloric Acid SCHEMBL7479212 0.99 ABCB11 (0.74) ABCB11OPRM1CYP2C19ADRA2ACYP2B6
Bromide SCHEMBL1402201 0.99 ABCB11 (0.74) ABCB11OPRM1CYP2C19ADRA2ACYP2B6
SCHEMBL3173500 0.99 ABCB11 (0.77) ABCB11OPRM1CYP2C19ADRA2ACYP2B6
SCHEMBL364610 0.99 ABCB11 (0.77) ABCB11OPRM1CYP2C19ADRA2ACYP2B6
SCHEMBL19148650 0.99 ABCB11 (0.77) ABCB11OPRM1CYP2C19ADRA2ACYP2B6
SCHEMBL30277249 0.99 ABCB11 (0.77) ABCB11OPRM1CYP2C19ADRA2ACYP2B6
SCHEMBL233523 0.99 ABCB11 (0.77) ABCB11OPRM1CYP2C19ADRA2ACYP2B6
SCHEMBL4770 0.99 ABCB11 (0.77) ABCB11OPRM1CYP2C19ADRA2ACYP2B6
SCHEMBL13403893 0.99 ABCB11 (0.77) ABCB11OPRM1CYP2C19ADRA2ACYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907397-B1 METHOD OF PREPARING CLOPIDOGREL AND INTERMEDIATES USED THEREIN HANMI HOLDINGS CO LTD (KR) 2011-06-29 EP disclosed
US-7763730-B2 Method preparation clopidogrel and intermediates used therein HANMI PHARM. CO., LTD (KR) 2010-07-27 US disclosed
US-7652140-B2 Method of preparing clopidogrel and intermediates used therein HANMI PHARM. CO., LTD (KR) 2010-01-26 US disclosed
US-20090318701-A1 METHOD PREPARATION CLOPIDOGREL AND INTERMEDIATES USED THEREIN HANMI PHARM CO., LTD. (KR) 2009-12-24 US disclosed
EP-1907397-A4 METHOD OF PREPARING CLOPIDOGREL AND INTERMEDIATES USED THEREIN HANMI PHARM IND CO LTD (KR) 2009-05-27 EP disclosed
US-20080214821-A1 Method of Preparing Clopidogrel and Intermediates Used Therein HANMI PHARM., CO., LTD. (KR) 2008-09-04 US disclosed
EP-1907397-A1 METHOD OF PREPARING CLOPIDOGREL AND INTERMEDIATES USED THEREIN Hanmi Pharm. Co., Ltd. (KR) 2008-04-09 EP disclosed
WO-2006137628-A1 METHOD OF PREPARING CLOPIDOGREL AND INTERMEDIATES USED THEREIN HANMI PHARM. CO., LTD. (KR) 2006-12-28 WO disclosed
US-4529596-A Anticoagulant; clopidogrel (Methyl Alpha -(4,5,6,7-tetrahydro-thieno(3,2-c)-5-pyridyl)-o-chlorophenyl-acetate) SANOFI, S.A. (FR) 1985-07-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090318701-A1 METHOD PREPARATION CLOPIDOGREL AND INTERMEDIATES USED THEREIN P2RY11, PTGIS, P2RY13 OPRM1 620/4885ADRA2A 324/4885OPRK1 1029/4885
US-20080214821-A1 Method of Preparing Clopidogrel and Intermediates Used Therein P2RY11, PTGIS, PTGIR OPRM1 632/4885ADRA2A 373/4885OPRK1 1117/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.