SCHEMBL19976942

SCHEMBL19976942

COc1ccc(F)cc1NC(=O)C(C)NC(=O)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.52
KMT2A Q03164 4/20 0.52
MAPT P10636 1/20 0.52
HTT P42858 1/20 0.52
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
HDAC1 Q13547 1/20 0.51
HDAC8 Q9BY41 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
CRHBP P24387 1/20 0.50
CRHR2 Q13324 1/20 0.50
KDM4E B2RXH2 2/20 0.49
ALDH1A1 P00352 1/20 0.49
CYP1A2 P05177 1/20 0.49
LMNA P02545 1/20 0.48
IRAK4 Q9NWZ3 1/20 0.47
GPR139 Q6DWJ6 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19976980 0.87 NPC1 (0.66) MEN1KMT2AMAPTHTTNPC1
SCHEMBL19977009 0.86 KMT2A (0.53) MEN1KMT2AMAPTHTTNPC1
SCHEMBL19976930 0.85 ALDH1A1 (0.55) MEN1KMT2AMAPTHTTCRHBP
SCHEMBL19976950 0.84 ALDH1A1 (0.51) MEN1KMT2AMAPTHTTNPC1
SCHEMBL16993955 0.83 PSMB5 (0.55) HDAC1HDAC8HDAC6ALDH1A1GPR139
SCHEMBL19977059 0.82 KMT2A (0.58) MEN1KMT2AMAPTNPC1RAB9A
SCHEMBL19976970 0.81 NPC1 (0.53) MEN1KMT2AMAPTHTTNPC1
SCHEMBL16999801 0.80 CTSL (0.54) HDAC1HDAC8HDAC6ALDH1A1
SCHEMBL18261135 0.80 CTSL (0.54) HDAC1HDAC8HDAC6ALDH1A1
SCHEMBL19976935 0.77 TUBB4A (0.47) MEN1KMT2AMAPTHTTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9919998-B2 Antibacterial agents: Nα-aroyl-N-aryl-phenylalaninamides RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2018-03-20 US disclosed