SCHEMBL19977009

SCHEMBL19977009

COc1ccc(F)cc1NC(=O)C(C)NC(=O)c1ccccc1F

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 7/20 0.53
MEN1 O00255 5/20 0.53
MAPT P10636 3/20 0.53
HTT P42858 1/20 0.53
ALDH1A1 P00352 4/20 0.52
KDM4E B2RXH2 2/20 0.52
SMN1; SMN2 Q16637 3/20 0.51
NPC1 O15118 3/20 0.51
RAB9A P51151 3/20 0.50
LMNA P02545 1/20 0.50
TDP1 Q9NUW8 1/20 0.49
HPGD P15428 1/20 0.49
PYGL P06737 2/20 0.47
IRAK4 Q9NWZ3 1/20 0.47
POLB P06746 1/20 0.47
BLM P54132 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47
CRHBP P24387 1/20 0.46
CRHR2 Q13324 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19976990 0.91 KMT2A (0.60) KMT2AMEN1MAPTHTTALDH1A1
SCHEMBL19976930 0.90 ALDH1A1 (0.55) KMT2AMEN1MAPTHTTALDH1A1
SCHEMBL19977067 0.89 CRHBP (0.60) KMT2AMEN1MAPTALDH1A1KDM4E
SCHEMBL19976976 0.88 KMT2A (0.56) KMT2AMEN1HTTALDH1A1KDM4E
SCHEMBL19976942 0.86 MEN1 (0.52) KMT2AMEN1MAPTHTTALDH1A1
SCHEMBL19976943 0.85 KMT2A (0.48) KMT2AMEN1MAPTHTTALDH1A1
SCHEMBL19976954 0.84 KMT2A (0.53) KMT2AMEN1MAPTALDH1A1KDM4E
SCHEMBL16994002 0.83 PSMB5 (0.60) KMT2AMEN1MAPTHTTALDH1A1
SCHEMBL19976935 0.81 TUBB4A (0.47) KMT2AMEN1MAPTHTTALDH1A1
SCHEMBL16999794 0.81 PSMB5 (0.53) KMT2AMEN1MAPTHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9919998-B2 Antibacterial agents: Nα-aroyl-N-aryl-phenylalaninamides RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2018-03-20 US disclosed